SCHEMBL23979015

SCHEMBL23979015

C=C(NCc1cccc(F)c1)c1cc(Cl)c(C(=C)CC)c(Cl)c1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.44
P2RY12 Q9H244 1/20 0.39
PTPN7 P35236 2/20 0.39
DUSP3 P51452 2/20 0.39
CNR1 P21554 1/20 0.38
SRC P12931 1/20 0.38
MAPK1 P28482 1/20 0.37
RAB9A P51151 1/20 0.37
ANPEP P15144 1/20 0.37
KDM5A P29375 1/20 0.36
KDM4C Q9H3R0 1/20 0.36
KDM5B Q9UGL1 1/20 0.36
NTRK1 P04629 2/20 0.36
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
DPP4 P27487 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978863 0.88 NPC1 (0.41) RAB9A
SCHEMBL23978714 0.88 CYP19A1 (0.35) P2RY12
SCHEMBL23978881 0.85 MEN1 (0.50) PTPN7DUSP3
SCHEMBL23978902 0.79 EPHX2 (0.39) EPHX2P2RY12PTPN7DUSP3CNR1
SCHEMBL23979115 0.74 TXNRD1 (0.36) P2RY12
SCHEMBL23978777 0.74 ROCK2 (0.48) CNR1
SCHEMBL23978774 0.71 MEN1 (0.50) EPHX2SRCKDM5AKDM4CKDM5B
SCHEMBL23978773 0.71 EPHX2 (0.49) EPHX2P2RY12
SCHEMBL26507428 0.69 MMP13 (0.40)
SCHEMBL24242018 0.69 SRC (0.45) EPHX2PTPN7DUSP3SRCMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed