SCHEMBL23979023

SCHEMBL23979023

C=C(NCc1cccc(C#N)c1)c1cc(Cl)c(C(=O)CC)c(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ERCC1 P07992 1/20 0.45
ERCC4 Q92889 1/20 0.45
VNN1 O95497 4/20 0.43
ROCK2 O75116 5/20 0.42
CNR1 P21554 1/20 0.41
MAOA P21397 1/20 0.40
ROCK1 Q13464 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.39
CHRM3 P20309 1/20 0.38
KLKB1 P03952 1/20 0.38
KLK1 P06870 1/20 0.38
MEP1A Q16819 1/20 0.38
MEP1B Q16820 1/20 0.38
GSK3B P49841 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978777 0.83 ROCK2 (0.48) ERCC1ERCC4VNN1ROCK2CNR1
SCHEMBL23978781 0.77 MAOA (0.53) ERCC1ERCC4VNN1ROCK2CNR1
SCHEMBL23978780 0.76 ROCK2 (0.51) ERCC1ERCC4VNN1ROCK2MAOA
SCHEMBL19049391 0.75 ERCC1 (0.64) ERCC1ERCC4VNN1ROCK2MAOA
SCHEMBL23978714 0.74 CYP19A1 (0.35) CHRM3
SCHEMBL23978863 0.74 NPC1 (0.41)
SCHEMBL38654611 0.72 ERCC1 (0.59) ERCC1ERCC4VNN1ROCK2CNR1
SCHEMBL8645386 0.72 ERCC1 (0.59) ERCC1ERCC4VNN1ROCK2CNR1
SCHEMBL23979015 0.72 EPHX2 (0.44) CNR1
SCHEMBL3461756 0.71 ERCC1 (0.60) ERCC1ERCC4VNN1ROCK2CNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed