SCHEMBL23979116

SCHEMBL23979116

NC(=O)NC[C@H](NC(=O)c1c(Cl)cc(N2CC(c3ccccc3)C2)cc1Cl)C(=O)OCc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 2/20 0.39
CAPN1 P07384 1/20 0.38
CTSS P25774 1/20 0.38
TGM2 P21980 3/20 0.37
F13A1 P00488 2/20 0.37
TGM1 P22735 2/20 0.37
POLB P06746 2/20 0.37
ITGB1 P05556 1/20 0.36
ITGA5 P08648 1/20 0.36
ACE P12821 1/20 0.36
MAPT P10636 2/20 0.35
CASP3 P42574 1/20 0.35
CCR1 P32246 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TGM6 O95932 1/20 0.34
ITGAL P20701 1/20 0.34
KAT2B Q92831 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23978822 0.88 ITGA4 (0.45) ITGA4ITGB1ITGA5ITGAL
SCHEMBL23979136 0.88 ITGA4 (0.38) ITGA4TGM2F13A1TGM1POLB
SCHEMBL30083835 0.85 ITGA4 (0.34) ITGA4CAPN1CTSSTGM2F13A1
SCHEMBL24804252 0.84 EPHX2 (0.43)
SCHEMBL24805441 0.84 EPHX2 (0.43)
SCHEMBL23978823 0.82 ITGA4 (0.36) ITGA4TGM2F13A1TGM1POLB
SCHEMBL24803399 0.79 EPHX2 (0.41) ITGA4CAPN1CTSSTGM2F13A1
SCHEMBL24805438 0.79 EPHX2 (0.41) ITGA4CAPN1CTSSTGM2F13A1
SCHEMBL30083824 0.79 CAPN1 (0.37) ITGA4CAPN1CTSSTGM2F13A1
SCHEMBL23978784 0.78 ITGB2 (0.44) ITGA4MAPTTDP1ITGAL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed