SCHEMBL23979136

SCHEMBL23979136

NC(=O)NC[C@H](NC(=O)c1c(Cl)cc(C(=O)N2CC(c3ccccc3)C2)cc1Cl)C(=O)OCc1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.38
ITGB2 P05107 4/20 0.37
ICAM1 P05362 4/20 0.37
ITGAL P20701 4/20 0.37
ITGB1 P05556 2/20 0.37
ITGA5 P08648 2/20 0.37
ACLY P53396 1/20 0.37
ACE P12821 1/20 0.36
HSD11B1 P28845 1/20 0.36
F13A1 P00488 1/20 0.36
TGM2 P21980 1/20 0.36
TGM1 P22735 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
GLRA1 P23415 1/20 0.36
CCR1 P32246 1/20 0.36
POLB P06746 1/20 0.36
SPR P35270 1/20 0.35
CSF1R P07333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23979116 0.88 ITGA4 (0.39) ITGA4ITGALITGB1ITGA5ACE
SCHEMBL23978784 0.87 ITGB2 (0.44) ITGA4ITGB2ICAM1ITGALTDP1
SCHEMBL24803484 0.85 EPHX2 (0.42) ITGB2ICAM1ITGALTDP1
SCHEMBL30083845 0.85 EPHX2 (0.42) ITGB2ICAM1ITGALTDP1
SCHEMBL23978804 0.85 EPHX2 (0.42) ITGB2ICAM1ITGALTDP1
SCHEMBL24804256 0.85 EPHX2 (0.42) ITGB2ICAM1ITGALTDP1
SCHEMBL23978731 0.83 MAPT (0.51) ITGB2ICAM1ITGALTDP1
SCHEMBL23978696 0.77 TACR1 (0.46) POLB
SCHEMBL23978763 0.76 ITGB1 (0.46) ITGB1ITGA5ACEPOLB
SCHEMBL23978822 0.76 ITGA4 (0.45) ITGA4ITGB2ICAM1ITGALITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222789-A1 INHIBITORS OF ALPHA 2 BETA 1 INTEGRIN AND METHODS OF USE THEREOF THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2021-11-04 WO disclosed