SCHEMBL23982003

SCHEMBL23982003

CC(C)(C)OC(=O)N1CCNC(c2cccnc2)C1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 3/20 0.52
MAPK1 P28482 1/20 0.46
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
KDM4E B2RXH2 1/20 0.44
ALDH1A1 P00352 1/20 0.44
MAPT P10636 1/20 0.44
HIF1A Q16665 1/20 0.44
CHRNB2 P17787 3/20 0.43
CHRNA4 P43681 3/20 0.43
CHRNA7 P36544 2/20 0.43
NAMPT P43490 1/20 0.43
KIT P10721 1/20 0.43
GBA1 P04062 1/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C19 P33261 2/20 0.42
POLB P06746 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2A6 P11509 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL38661093 0.87 MAPK1 (0.45) GPR119MAPK1CYP2D6CYP2C9GRM1
SCHEMBL23982034 0.87 GPR119 (0.43) GPR119MAPK1KDM4EMAPT
SCHEMBL940218 0.87 MAPK1 (0.50) GPR119MAPK1KDM4E
SCHEMBL28225677 0.87 MAPK1 (0.50) GPR119MAPK1KDM4E
SCHEMBL5651780 0.87 MAPK1 (0.50) GPR119MAPK1KDM4E
SCHEMBL19745334 0.87 MAPK1 (0.50) GPR119MAPK1KDM4E
Hydrochloric Acid SCHEMBL28503227 0.85 MAPK1 (0.49) GPR119MAPK1KDM4E
SCHEMBL30273306 0.82 STS (0.40) GPR119MAPK1MEN1KMT2AKDM4E
SCHEMBL23981737 0.82 STS (0.40) GPR119MAPK1MEN1KMT2AKDM4E
SCHEMBL15365495 0.81 ESR2 (0.44) GPR119MAPK1KDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2026101698-A1 HEPCIDIN MIMETIC COMPOUNDS AND USES THEREOF PROTAGONIST THERAPEUTICS, INC. (US) 2026-05-15 WO disclosed
CN-122036605-A Antagonists of GPR39 proteins 俄勒冈健康科学大学 2026-05-15 CN disclosed
CN-117794525-A Anticancer compounds 加利福尼亚大学董事会 2024-03-29 CN disclosed
US-20230174484-A1 ANTAGONISTS OF GPR39 PROTEIN UNIV OREGON HEALTH & SCIENCE (US) 2023-06-08 US disclosed
US-20230174484-A1 ANTAGONISTS OF GPR39 PROTEIN UNIV OREGON HEALTH & SCIENCE (US) 2023-06-08 US disclosed
US-20230174484-A1 ANTAGONISTS OF GPR39 PROTEIN UNIV OREGON HEALTH & SCIENCE (US) 2023-06-08 US disclosed
CN-115996908-A Antagonists of GPR39 proteins 俄勒冈健康科学大学 2023-04-21 CN disclosed
WO-2021222858-A1 ANTAGONISTS OF GPR39 PROTEIN OREGON HEALTH & SCIENCE UNIVERSITY (US) 2021-11-04 WO disclosed
CN-107253963-A Pyridone and azepine pyridinone compounds and application method 吉利德康涅狄格有限公司 2017-10-17 CN disclosed
CN-107011348-A It is used as the heteroaryl pyridines ketone and azepine pyridinone compounds of the inhibitor of BTK activity 霍夫曼-拉罗奇有限公司 2017-08-04 CN disclosed
CN-103038233-B Pyridone and azapyridone compounds and methods of use 吉利德康涅狄格有限公司 2017-06-20 CN disclosed
CN-104125959-B Heteroaryl pyridone and aza-pyridone compounds as inhibitors of BTK activity 霍夫曼-拉罗奇有限公司 2017-05-03 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174484-A1 ANTAGONISTS OF GPR39 PROTEIN GPR39, GPR139, GPR119 GPR119 3/4885MAPK1 3174/4885MEN1 3377/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.