Tyrphostin 25

Tyrphostin 25

SCHEMBL239879

N#CC(C#N)=Cc1cc(O)c(O)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 10/20 1.00
MEN1 O00255 8/20 1.00
KMT2A Q03164 8/20 1.00
MAPT P10636 8/20 1.00
ALDH1A1 P00352 7/20 1.00
HPGD P15428 6/20 1.00
BLM P54132 6/20 1.00
LMNA P02545 6/20 1.00
KDM4E B2RXH2 6/20 1.00
CYP3A4 P08684 5/20 1.00
CYP2C9 P11712 5/20 1.00
HSD17B10 Q99714 5/20 1.00
ALOX15 P16050 4/20 1.00
NFKB1 P19838 4/20 1.00
PMP22 Q01453 4/20 1.00
SMN1; SMN2 Q16637 4/20 1.00
HIF1A Q16665 4/20 1.00
TDP1 Q9NUW8 4/20 1.00
RGS12 O14924 3/20 1.00
GNAI1 P63096 3/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10144263 0.88 EGFR (0.78) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL10186359 0.86 EGFR (1.00) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL8485552 0.86 EGFR (0.75) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL29457559 0.83 EGFR (1.00) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL3459584 0.83 EGFR (1.00) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL12617223 0.83 EGFR (0.70) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL31618898 0.79 ALDH1A1 (1.00) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL10144550 0.79 ALDH1A1 (1.00) EGFRMEN1KMT2AMAPTALDH1A1
SCHEMBL8609619 0.79 EGFR (1.00) EGFRMEN1KMT2AMAPTALDH1A1
Tyrphostin 23 SCHEMBL241922 0.78 EGFR (1.00) EGFRMEN1KMT2AMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 477 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4577832-A1 METHOD FOR PREDICTING THE RESPONSE TO AN INHIBITOR OF EGFR KINASE ACTIVITY Indivumed GmbH (DE) 2025-07-02 EP claimed
WO-2024042077-A1 METHOD FOR PREDICTING THE RESPONSE TO AN INHIBITOR OF EGFR KINASE ACTIVITY INDIVUMED GMBH (DE) 2024-02-29 WO claimed
CN-116660543-A Diagnostic and prognostic markers for nonalcoholic fatty liver disease and uses thereof 中国人民解放军陆军军医大学第一附属医院 2023-08-29 CN claimed
EP-2516626-B1 DIFFERENTIATION OF HUMAN EMBRYONIC STEM CELLS JANSSEN BIOTECH INC (US) 2017-05-10 EP claimed
US-9133439-B2 Differentiation of human embryonic stem cells JANSSEN BIOTECH, INC. (US) 2015-09-15 US claimed
EP-2516626-A2 DIFFERENTIATION OF HUMAN EMBRYONIC STEM CELLS Janssen Biotech, Inc. (US) 2012-10-31 EP claimed
CN-102712902-A Differentiation of human embryonic stem cells CENTOCOR ORTHO BIOTECH INC 2012-10-03 CN claimed
US-20120076781-A1 METHODS OF TREATING CANCERS WITH HER3 ANTISENSE OLIGONUCLEOTIDES SANTARIS PHARMA A/S (DK) 2012-03-29 US claimed
EP-2419110-A1 METHODS OF TREATING CANCERS WITH HER3 ANTISENSE OLIGONUCLEOTIDES Enzon Pharmaceuticals, Inc. (US) 2012-02-22 EP claimed
US-20120004285-A1 ERBB-3 (HER3)-SELECTIVE COMBINATION THERAPY ENZON PHARMACEUTICALS, INC. (US) 2012-01-05 US claimed
US-20080286670-A1 Photoconductors containing charge transport chelating components XEROX CORPORATION 2008-11-20 US claimed
WO-2007106432-A2 EGF RECEPTOR PHOSPHORYLATION STATUS FOR DISEASE TREATMENT GEORGE MASON INTELLECTUAL PROPERTIES, INC. (US) 2007-09-20 WO claimed
US-7052692-B1 Role of tyrosine phosphorylation of a cellular protein in adeno-associated virus 2-mediated transgene expression ADVANCED RESEARCH & TECHNOLOGY INSTITUTE (US) 2006-05-30 US claimed
EP-1156775-B1 REDUCTION OF HAIR GROWTH GILLETTE CO (US) 2006-05-17 EP claimed
EP-1156775-A1 REDUCTION OF HAIR GROWTH THE GILLETTE COMPANY (US) 2001-11-28 EP claimed
US-6121269-A TOPICALLY APPLYING A PROTEIN-TYROSINE KINASE INHIBITOR TO SKIN TO REDUCE ANDROGEN-STIMULATED HAIR GROWTH WITHOUT SIDE EFFECTS GILLETTE COMPANY, THE, A DELAWARE CORPORATION 2000-09-19 US claimed
WO-2000050002-A1 REDUCTION OF HAIR GROWTH THE GILLETTE COMPANY (US) 2000-08-31 WO claimed
EP-0614661-A2 Benzylidene- and cinnamylidine-malononitrile derivatives for the inhibition of proliferative processes in mammalian cells YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1994-09-14 EP claimed
EP-0403238-A2 Cosmetic composition UNILEVER PLC (GB) 1990-12-19 EP claimed
EP-0322738-A2 Benzylidene-malononitrile derivatives for the inhibition of proliferative processes in mammalian cells YISSUM RESEARCH DEVELOPMENT COMPANY OF THE HEBREW UNIVERSITY OF JERUSALEM (IL) 1989-07-05 EP claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120076781-A1 METHODS OF TREATING CANCERS WITH HER3 ANTISENSE OLIGONUCLEOTIDES ERBB3, ERBB2, EGFR EGFR 3/4885MEN1 2801/4885KMT2A 1292/4885
US-20120004285-A1 ERBB-3 (HER3)-SELECTIVE COMBINATION THERAPY ERBB3, ERBB2, EGFR EGFR 3/4885MEN1 2296/4885KMT2A 2276/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.