SCHEMBL24007286

SCHEMBL24007286

Cc1cc(F)ccc1C(C)NN

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SOS1 Q07889 4/20 0.36
GPR139 Q6DWJ6 1/20 0.34
HTR2A P28223 2/20 0.33
SLC6A4 P31645 2/20 0.33
KCNH2 Q12809 2/20 0.33
CYP2D6 P10635 1/20 0.32
POLB P06746 1/20 0.32
ALDH1A1 P00352 2/20 0.31
HDAC4 P56524 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18280637 0.78 PDE2A (0.44) HTR2AALDH1A1
SCHEMBL25688856 0.78 PDE2A (0.44) HTR2AALDH1A1
SCHEMBL29074414 0.78 GPR139 (0.41) SOS1GPR139POLB
SCHEMBL84044 0.77 ALDH1A1 (0.41) ALDH1A1
Hydrochloric Acid SCHEMBL29074379 0.76 GPR139 (0.40) SOS1GPR139POLB
Hydrochloric Acid SCHEMBL31561502 0.76 PDE2A (0.43) HTR2AALDH1A1
Hydrochloric Acid SCHEMBL19205712 0.76 PDE2A (0.43) HTR2AALDH1A1
Hydrochloric Acid SCHEMBL18449678 0.76 PDE2A (0.43) HTR2AALDH1A1
SCHEMBL25373380 0.74 PTGS1 (0.32) HTR2ACYP2D6ALDH1A1
SCHEMBL21323637 0.74 ACHE (0.33) SOS1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021226208-A2 HETEROAROMATIC MACROCYCLIC ETHER CHEMOTHERAPEUTIC AGENTS NUVALENT, INC. (US) 2021-11-11 WO disclosed