SCHEMBL24015809

SCHEMBL24015809

Cc1sc(C(F)(F)F)nc1N

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
NOS1 P29475 1/20 0.34
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
MPL P40238 2/20 0.33
HSP90AA1 P07900 1/20 0.32
HSP90AB1 P08238 1/20 0.32
PRMT6 Q96LA8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13841474 0.76 NOS1 (0.42) ALDH1A1NOS1
SCHEMBL26747517 0.74 COMT (0.33) ALDH1A1
SCHEMBL22121867 0.73 ALDH1A1 (0.32) ALDH1A1
SCHEMBL24015810 0.73 ALDH1A1 (0.41) ALDH1A1NOS1HPGDHSD17B10HSP90AA1
SCHEMBL5627523 0.73
SCHEMBL23942114 0.68
SCHEMBL8627226 0.67
SCHEMBL2616831 0.67
SCHEMBL23354329 0.67 RBP4 (0.39) ALDH1A1HPGD
SCHEMBL23371356 0.66 GAA (0.33) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023078813-A1 HETEROBIFUNCTIONAL MOLECULES AS TEAD INHIBITORS MERCK PATENT GMBH (DE) 2023-05-11 WO disclosed
WO-2021224291-A1 TRICYCLIC HETEROCYCLES USEFUL AS TEAD BINDERS MERCK PATENT GMBH (DE) 2021-11-11 WO disclosed