SCHEMBL24036748

SCHEMBL24036748

COC(=O)CC(NC(=O)CNC(=O)OC(C)(C)C)c1cccc(C2CC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA1B Q00975 2/20 0.38
EPHX2 P34913 1/20 0.36
GPR139 Q6DWJ6 2/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
ROCK2 O75116 2/20 0.35
PRKG1 Q13976 1/20 0.35
CCR2 P41597 1/20 0.34
PTPRB P23467 1/20 0.34
REN P00797 1/20 0.34
PPARG P37231 1/20 0.33
RAB9A P51151 1/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25624750 1.00 CACNA1B (0.38) CACNA1BEPHX2GPR139CTSSCTSK
SCHEMBL27406042 0.90 CACNA1B (0.43) CACNA1BCTSSCTSKROCK2PRKG1
SCHEMBL29861275 0.90 CACNA1B (0.43) CACNA1BCTSSCTSKROCK2PRKG1
SCHEMBL24036823 0.85 CACNA1B (0.41) CACNA1BEPHX2GPR139CTSSCTSK
SCHEMBL25624830 0.85 GPR139 (0.42) EPHX2GPR139CTSSCTSKPTPRB
SCHEMBL24036832 0.84 WDR5 (0.44) EPHX2GPR139CTSSCTSKPTPRB
SCHEMBL24036746 0.84 GPR139 (0.39) EPHX2GPR139CTSSCTSKPTPRB
SCHEMBL25753975 0.84 EGFR (0.43) EPHX2GPR139CTSSCTSKHDAC3
SCHEMBL24036744 0.82 ITGB3 (0.40) CACNA1BEPHX2GPR139CTSSCTSK
SCHEMBL24036747 0.82 GPR139 (0.46) GPR139CTSSCTSKHDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021230325-A1 1, 4, 5, 6-TETRAHYDROPYRIMIDINE-2-AMINE DERIVATIVE 宇部興産株式会社 2021-11-18 WO disclosed