SCHEMBL2404077

SCHEMBL2404077

COc1cc(CC(=O)N(C)C2CC2)ccc1O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.58
TSHR P16473 2/20 0.58
GAA P10253 1/20 0.58
NFKB1 P19838 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
CCR5 P51681 1/20 0.53
KDM4E B2RXH2 1/20 0.48
ALOX5 P09917 1/20 0.48
OR51E2 Q9H255 1/20 0.48
SHBG P04278 2/20 0.47
TAAR1 Q96RJ0 2/20 0.47
MAPK1 P28482 1/20 0.47
FOS P01100 1/20 0.46
TTR P02766 1/20 0.46
JUN P05412 1/20 0.46
NR3C1 P04150 1/20 0.46
HSD17B1 P14061 1/20 0.46
HSD17B2 P37059 1/20 0.46
LMNA P02545 1/20 0.46
GLA P06280 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2403525 0.89 CCR5 (0.64) ALDH1A1GAACCR5LMNA
SCHEMBL2405228 0.84 CCR5 (0.57) ALDH1A1TSHRCCR5KDM4EMAPK1
SCHEMBL2404781 0.84 CCR5 (0.57) ALDH1A1CCR5KDM4EMAPK1LMNA
SCHEMBL2406042 0.84 CCR5 (0.53) ALDH1A1GAACCR5
SCHEMBL2403861 0.82 SIGMAR1 (0.62) ALDH1A1GAACCR5MAPK1
SCHEMBL2405481 0.82 CCR5 (0.52) ALDH1A1GAACCR5LMNA
SCHEMBL2406179 0.81 CCR5 (0.57) ALDH1A1TSHRTDP1CCR5MAPK1
SCHEMBL2410390 0.81 CCR5 (0.57) ALDH1A1TSHRTDP1CCR5MAPK1
SCHEMBL29066070 0.80 TSHR (0.65) ALDH1A1TSHRGAANFKB1TDP1
SCHEMBL9028072 0.80 ALDH1A1 (0.48) ALDH1A1TSHRGAANFKB1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES ACTELION PHARMACEUTICALS LTD. (CH) 2011-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212968-A1 PHENETHYLAMIDE DERIVATIVES AND THEIR HETEROCYCLIC ANALOGUES HCRTR2, HCRTR1, HRH3 ALDH1A1 2292/4885TSHR 289/4885GAA 2389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.