SCHEMBL2406362

SCHEMBL2406362

Clc1ccc2c(-c3ncc[nH]3)c[nH]c2c1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 2/20 0.56
GSK3B P49841 1/20 0.55
GPR84 Q9NQS5 1/20 0.46
ALDH1A1 P00352 1/20 0.44
IDH1 O75874 1/20 0.43
MDM2 Q00987 3/20 0.42
MDM4 O15151 2/20 0.42
TP53 P04637 2/20 0.42
MAP3K14 Q99558 1/20 0.42
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
SLC6A4 P31645 1/20 0.40
TDO2 P48775 2/20 0.40
NR4A2 P43354 1/20 0.39
IMPDH2 P12268 2/20 0.38
ALOX5 P09917 1/20 0.38
ELANE P08246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1325544 0.77 HSD17B10 (0.54) DYRK1AGSK3BALDH1A1MAP3K14ADRA1A
SCHEMBL3631532 0.76 RAB9A (0.50) GSK3BALDH1A1
SCHEMBL31429694 0.75 IDO1 (0.51) ALDH1A1
SCHEMBL8542466 0.75 ALDH1A1 (0.49) GSK3BALDH1A1
SCHEMBL8537063 0.73 NR4A2 (0.43) ALDH1A1TP53NR4A2
SCHEMBL31429733 0.73 IDO1 (0.58) ALDH1A1
SCHEMBL29084865 0.73 IDO1 (0.58) ALDH1A1
SCHEMBL8541383 0.73 KMO (0.43) GSK3BALDH1A1
SCHEMBL28379218 0.73 DYRK1A (0.75) DYRK1AGSK3BGPR84MAP3K14ALOX5
SCHEMBL8558526 0.72 NPC1 (0.40) GSK3BALDH1A1NR4A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011106650-A2 NOVEL P53-MDM2/P53-MDM4 ANTAGONISTS TO TREAT PROLIFERATIVE DISEASE UNIVERSITY OF PITTSBURGH - OF THE COMMONWEALTH SYSTEM OF HIGHER EDUCATION (US) 2011-09-01 WO disclosed