SCHEMBL24070302

SCHEMBL24070302

COC(=O)c1c(Cl)cc(Cl)nc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.42
ALPL P05186 1/20 0.38
KMT2A Q03164 3/20 0.37
ALDH1A1 P00352 4/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
NPSR1 Q6W5P4 1/20 0.36
MAPT P10636 2/20 0.36
POLB P06746 1/20 0.36
MEN1 O00255 1/20 0.36
CASP3 P42574 1/20 0.36
SENP7 Q9BQF6 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
CA14 Q9ULX7 1/20 0.36
NQO2 P16083 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PLA2G2A P14555 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31388114 0.83 KDM4E (0.40) KDM4EALPLALDH1A1SMN1; SMN2NPSR1
SCHEMBL12380495 0.82 KDM4E (0.44) KDM4EKMT2AALDH1A1SMN1; SMN2NPSR1
SCHEMBL1710208 0.82 KDM4E (0.44) KDM4EKMT2AALDH1A1SMN1; SMN2NPSR1
SCHEMBL29364806 0.79 NQO2 (0.44) KDM4EKMT2AALDH1A1SMN1; SMN2NPSR1
SCHEMBL145259 0.79 NQO2 (0.44) KDM4EKMT2AALDH1A1SMN1; SMN2NPSR1
SCHEMBL1327502 0.79 GABRP (0.40) KDM4EALDH1A1SMN1; SMN2MAPTL3MBTL1
SCHEMBL24069421 0.78 ALDH1A1 (0.44) KDM4EALPLKMT2AALDH1A1SMN1; SMN2
SCHEMBL17054798 0.77 KDM4E (0.40) KDM4EKMT2AALDH1A1SMN1; SMN2NPSR1
SCHEMBL22623064 0.77 POLB (0.42) KMT2AALDH1A1SMN1; SMN2MAPTPOLB
SCHEMBL5788599 0.76 CA12 (0.42) KDM4EALPLKMT2AALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115551867-B Fused tricyclic compounds, pharmaceutical compositions and uses thereof 劲方医药科技(上海)有限公司 2024-02-20 CN disclosed
US-20230203060-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF GENFLEET THERAPEUTICS (SHANGHAI) INC. (CN) 2023-06-29 US disclosed
US-20230203060-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF GENFLEET THERAPEUTICS (SHANGHAI) INC. (CN) 2023-06-29 US disclosed
CN-115551867-A Fused tricyclic compound, pharmaceutical composition and application thereof 劲方医药科技(上海)有限公司 2022-12-30 CN disclosed
WO-2021239058-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF 劲方医药科技(上海)有限公司 2021-12-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230203060-A1 FUSED TRICYCLIC COMPOUND, PHARMACEUTICAL COMPOSITION THEREOF, AND USE THEREOF KRAS, NRAS, TP53 KDM4E 4302/4885ALPL 3873/4885KMT2A 3065/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.