SCHEMBL2407643

SCHEMBL2407643

COc1cccc(S(=O)(=O)n2cc(CN(C)C(=O)OC(C)(C)C)cc2Br)c1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM5 P08912 1/20 0.42
USP2 O75604 1/20 0.42
HTR6 P50406 6/20 0.40
PTGER2 P43116 1/20 0.40
ALDH1A1 P00352 1/20 0.39
PKM P14618 1/20 0.39
HDAC1 Q13547 1/20 0.38
MEP1B Q16820 1/20 0.38
MET P08581 1/20 0.37
LIMK2 P53671 1/20 0.37
TAS2R14 Q9NYV8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31754855 0.90 F2 (0.37) CHRM5USP2HTR6PTGER2PKM
SCHEMBL1157010 0.89 HTR6 (0.41) CHRM5HTR6ALDH1A1PKM
SCHEMBL30089413 0.88 HTR2C (0.36) HTR6PKMHDAC1
SCHEMBL1156487 0.88 HTR2C (0.36) HDAC1MET
SCHEMBL30089406 0.88 F2 (0.37) CHRM5USP2HTR6PTGER2ALDH1A1
SCHEMBL1156621 0.88 HTR2C (0.42) HTR6
SCHEMBL31755377 0.87 SMPD1 (0.37) HTR6ALDH1A1
SCHEMBL1156562 0.87 HTR6 (0.40) HTR6ALDH1A1
SCHEMBL2416549 0.87 RIPK1 (0.39) HTR6ALDH1A1PKM
SCHEMBL30089348 0.87 HTR6 (0.40) HTR6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118894801-A Pyrrole sulfonyl derivative, and preparation method and application thereof 天地恒一制药股份有限公司 2024-11-05 CN disclosed
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed