SCHEMBL2408052

SCHEMBL2408052

O=C(c1ccc(-c2ccccc2)cc1)N1CCc2ncnc(Cl)c2C1

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 2/20 0.57
KCNK9 Q9NPC2 1/20 0.57
MTHFD2 P13995 6/20 0.50
P2RX7 Q99572 2/20 0.48
MAPK1 P28482 2/20 0.48
HPGD P15428 1/20 0.48
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SLC6A7 Q99884 3/20 0.46
ALDH1A1 P00352 2/20 0.46
TSHR P16473 1/20 0.46
POLB P06746 2/20 0.45
L3MBTL1 Q9Y468 1/20 0.44
TRPV1 Q8NER1 1/20 0.44
MGLL Q99685 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12321175 0.87 KCNK3 (0.58) KCNK3KCNK9MTHFD2P2RX7MAPK1
SCHEMBL12320789 0.86 KCNK3 (0.60) KCNK3KCNK9MTHFD2MAPK1HPGD
SCHEMBL12321214 0.79 MTHFD2 (0.61) KCNK3KCNK9MTHFD2MAPK1HPGD
SCHEMBL2471575 0.77 KCNK3 (0.65) KCNK3KCNK9MTHFD2MEN1KMT2A
SCHEMBL12321215 0.77 KCNK3 (0.60) KCNK3KCNK9MTHFD2MAPK1SLC6A7
SCHEMBL12320843 0.76 KCNK3 (0.55) KCNK3KCNK9MTHFD2MAPK1HPGD
SCHEMBL2410631 0.76 KCNK3 (0.59) KCNK3KCNK9MTHFD2MAPK1HPGD
SCHEMBL2410232 0.76 KCNK3 (0.72) KCNK3KCNK9MTHFD2HPGDMEN1
SCHEMBL2410478 0.76 KCNK3 (0.73) KCNK3KCNK9MTHFD2MAPK1MEN1
SCHEMBL12320841 0.76 SLC6A7 (0.66) KCNK3KCNK9MTHFD2MAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011103715-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed
WO-2011106276-A1 TASK CHANNEL ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2011-09-01 WO disclosed