SCHEMBL24089908

SCHEMBL24089908

O=c1c2cc(F)ccc2nc(Nc2cccc(CN3CCC3)c2)n1-c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ACP1 P24666 5/20 0.45
IDO1 P14902 3/20 0.43
TDO2 P48775 3/20 0.43
IDO2 Q6ZQW0 3/20 0.43
HTR7 P34969 3/20 0.43
KCNH2 Q12809 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
AVPR1B P47901 3/20 0.42
FAAH O00519 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23065101 0.90 MEN1 (0.48) ALDH1A1MEN1KMT2AHSD17B10ACP1
SCHEMBL24089906 0.89 ACP1 (0.50) ALDH1A1MEN1KMT2AHSD17B10ACP1
SCHEMBL24090101 0.89 ACP1 (0.51) ALDH1A1ACP1AVPR1BFAAHSMN1; SMN2
SCHEMBL29623188 0.88 MEN1 (0.52) ALDH1A1MEN1KMT2AHSD17B10ACP1
SCHEMBL23065098 0.88 MEN1 (0.52) ALDH1A1MEN1KMT2AHSD17B10ACP1
SCHEMBL29623301 0.86 TOP2A (0.48) ALDH1A1TDO2IDO2HTR7
SCHEMBL24089966 0.86 TOP2A (0.48) ALDH1A1TDO2IDO2HTR7
SCHEMBL24090098 0.83 TDO2 (0.49) ALDH1A1ACP1IDO1TDO2IDO2
SCHEMBL23045334 0.82 TDO2 (0.50) IDO1TDO2IDO2HTR7SMN1; SMN2
SCHEMBL29623155 0.82 TDO2 (0.50) IDO1TDO2IDO2HTR7SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114650986-A 2-aminoquinazolinone derivatives 住友制药株式会社 2022-06-21 CN claimed
CN-114650986-A 2-aminoquinazolinone derivatives 住友制药株式会社 2022-06-21 CN disclosed
US-11352366-B2 2-aminoquinazolinone derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-06-07 US disclosed
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-05-12 US disclosed
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220143020-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, CRKL ALDH1A1 645/4885MEN1 1124/4885KMT2A 1257/4885
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, SLC26A3 ALDH1A1 739/4885MEN1 1282/4885KMT2A 967/4885
US-11352366-B2 2-aminoquinazolinone derivative CNKSR1, HAX1, SLC26A3 ALDH1A1 739/4885MEN1 1282/4885KMT2A 967/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.