SCHEMBL2409035

SCHEMBL2409035

CN(Cc1cn(S(=O)(=O)c2cccc(CCl)c2)c(-c2cccnc2F)c1F)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.35
SLC6A4 P31645 6/20 0.35
RXFP1 Q9HBX9 1/20 0.35
KAT8 Q9H7Z6 2/20 0.34
F2 P00734 4/20 0.32
KAT6A Q92794 2/20 0.32
KAT5 Q92993 2/20 0.32
HTR2A P28223 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
GLS O94925 1/20 0.31
PDK2 Q15119 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2415887 0.94 HTR2C (0.34) HTR2CSLC6A4RXFP1KAT8F2
SCHEMBL2411933 0.92 HTR2C (0.33) HTR2CSLC6A4RXFP1KAT8F2
SCHEMBL2408489 0.92 HTR2C (0.36) HTR2CSLC6A4RXFP1KAT8F2
SCHEMBL4420269 0.91 HTR6 (0.37) HTR2CSLC6A4KAT8F2HTR2A
SCHEMBL2407588 0.90 MET (0.38) HTR2CSLC6A4KAT8F2KAT6A
SCHEMBL2409254 0.89 F2 (0.34) HTR2CSLC6A4KAT8F2HTR2A
SCHEMBL2411540 0.89 MET (0.41) F2
SCHEMBL5002713 0.88 RXFP1 (0.35) RXFP1MEN1KMT2A
SCHEMBL2408606 0.88 TDP1 (0.37) HTR2CSLC6A4RXFP1MEN1KMT2A
SCHEMBL2410115 0.88 RORC (0.38) KAT8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed