SCHEMBL2409151

SCHEMBL2409151

CC(=O)c1cccc(S(=O)(=O)n2cc(CC(NC(=O)O)C(C)(C)C)cc2-c2cccnc2F)c1

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CHRM5 P08912 1/20 0.32
PDE4A P27815 1/20 0.32
KCNH2 Q12809 1/20 0.32
NAMPT P43490 1/20 0.31
GAA P10253 1/20 0.31
HTT P42858 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
ADAMTS4 O75173 1/20 0.31
PKM P14618 1/20 0.31
TSHR P16473 1/20 0.31
PTGDR2 Q9Y5Y4 2/20 0.31
CCKAR P32238 1/20 0.31
KMT2A Q03164 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2418766 0.92 PTGDR (0.35) ALDH1A1PKMTSHRPTGDR2KMT2A
SCHEMBL2415722 0.91 PTGDR2 (0.35) SMN1; SMN2PTGDR2CCKARKMT2A
SCHEMBL2412871 0.88 PTGDR2 (0.42) PDE4ANAMPTPTGDR2CCKAR
SCHEMBL1278109 0.88 FPR1 (0.34) ALDH1A1SMN1; SMN2GAATSHRPTGDR2
SCHEMBL2416815 0.88 GRM4 (0.33) ADAMTS4PKMPTGDR2CCKAR
SCHEMBL2414117 0.88 APLNR (0.36) NAMPTADAMTS4PTGDR2
SCHEMBL2412419 0.87 GRM4 (0.39) ALDH1A1SMN1; SMN2NAMPTNPSR1TSHR
SCHEMBL1278409 0.86 PTGDR2 (0.32) NAMPTPTGDR2CCKAR
SCHEMBL2412112 0.85 KAT6A (0.32) ALDH1A1SMN1; SMN2NAMPTTSHRPTGDR2
SCHEMBL2413126 0.85

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed