SCHEMBL24101686

SCHEMBL24101686

Cc1csc(NC(=O)Cc2csc(Nc3cccc(C(F)(F)F)c3)n2)n1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 1/20 0.63
MAPT P10636 11/20 0.58
CYP1A2 P05177 3/20 0.58
CYP3A4 P08684 3/20 0.58
CYP2D6 P10635 3/20 0.58
CYP2C9 P11712 3/20 0.58
CYP2C19 P33261 3/20 0.58
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
LMNA P02545 2/20 0.58
NPSR1 Q6W5P4 3/20 0.58
HPGD P15428 1/20 0.58
HTT P42858 1/20 0.58
GPR35 Q9HC97 1/20 0.58
ALDH1A1 P00352 3/20 0.57
UBE2N P61088 1/20 0.56
GAA P10253 3/20 0.54
RORC P51449 1/20 0.52
KDM4E B2RXH2 2/20 0.50
MAPK1 P28482 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14069823 0.84 MAPT (0.59) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL11516149 0.83 PDE5A (0.64) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL11517104 0.82 PDE5A (0.62) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL11519026 0.82 PDE5A (0.62) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL11516869 0.82 PDE5A (0.62) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL24101688 0.80 NPC1 (0.68) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL10464324 0.78 VCP (0.58) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL11515699 0.78 PDE5A (0.57) PDE5AMAPTCYP1A2CYP3A4CYP2D6
SCHEMBL4876936 0.76 VCP (0.61) MAPTCYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL24101768 0.76 MAPT (0.79) MAPTMEN1KMT2ALMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021249517-A1 A MOLECULAR GLUE REGULATING CDK12-DDB1 INTERACTION TO TRIGGER CYCLIN K DEGRADATION NATIONAL INSTITUTE OF BIOLOGICAL SCIENCES, BEIJING (CN) 2021-12-16 WO disclosed