SCHEMBL24123763

SCHEMBL24123763

CC(C)c1ccc(N2CC(N(C)C)C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.42
L3MBTL1 Q9Y468 2/20 0.41
NOTUM Q6P988 2/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
MGLL Q99685 1/20 0.39
HTR2A P28223 1/20 0.38
HTR2C P28335 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
MAPK1 P28482 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
GAA P10253 1/20 0.37
ALOX15 P16050 1/20 0.37
ALOX12 P18054 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
HPGD P15428 1/20 0.37
ACACB O00763 1/20 0.36
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14923971 0.86 RORC (0.47) HRH3HTR2AHTR2CACACBRORC
SCHEMBL16451234 0.82 HRH3 (0.47) HRH3L3MBTL1MEN1KMT2AHTR2A
SCHEMBL189433 0.81 MAPT (0.47) HRH3L3MBTL1MEN1KMT2AALDH1A1
SCHEMBL24123779 0.79 ADRB1 (0.44) HRH3L3MBTL1NOTUMMEN1KMT2A
SCHEMBL26498514 0.78 L3MBTL1 (0.41) HRH3L3MBTL1NOTUMMEN1KMT2A
SCHEMBL12499527 0.77 HRH3 (0.37) HRH3MGLLHTR2AHTR2CRORC
SCHEMBL24352426 0.77 L3MBTL1 (0.43) HRH3L3MBTL1NOTUMMEN1KMT2A
SCHEMBL22854281 0.77 L3MBTL1 (0.43) HRH3L3MBTL1NOTUMMEN1KMT2A
SCHEMBL30206343 0.77 MCHR1 (0.37) HRH3HTR2AHTR2C
SCHEMBL30493024 0.76 DDB1 (0.49) HRH3NOTUMMEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021254389-A1 PYRAZOLO[3,4-D]PYRIMIDINE-3-KETONE DERIVATIVE AS WEE-1 INHIBITOR 微境生物医药科技(上海)有限公司 2021-12-23 WO disclosed