SCHEMBL24136384

SCHEMBL24136384

N=C/C(Br)=C\NCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADH1B P00325 1/20 0.47
ADH1C P00326 1/20 0.47
ADH1A P07327 1/20 0.47
ADH7 P40394 1/20 0.47
ALOX12 P18054 3/20 0.42
ALDH1A1 P00352 3/20 0.42
HPGD P15428 2/20 0.42
IDO1 P14902 2/20 0.42
THRB P10828 1/20 0.42
MAPT P10636 5/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
POLB P06746 1/20 0.41
GAA P10253 1/20 0.41
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
NR4A1 P22736 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP2C9 P11712 1/20 0.37
CYP3A4 P08684 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24014177 0.78 ALDH1A1 (0.50) ALOX12ALDH1A1HPGDMAPTMEN1
SCHEMBL16903733 0.78 ADH1B (0.47) ADH1BADH1CADH1AADH7ALOX12
SCHEMBL15075659 0.76 ADH1B (0.46) ADH1BADH1CADH1AADH7ALOX12
SCHEMBL21095906 0.75 ADH1B (0.44) ADH1BADH1CADH1AADH7ALOX12
SCHEMBL10151057 0.75 ADH1B (0.53) ADH1BADH1CADH1AADH7ALOX12
SCHEMBL21095759 0.75 ADH1B (0.44) ADH1BADH1CADH1AADH7ALOX12
SCHEMBL21210266 0.74 ADH1B (0.43) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL3084417 0.73 ADH1B (0.60) ADH1BADH1CADH1AADH7ALOX12
SCHEMBL20344648 0.73 ADH1B (0.46) ADH1BADH1CADH1AADH7ALDH1A1
SCHEMBL627479 0.72 ADH1B (0.54) ADH1BADH1CADH1AADH7ALOX12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023165943-A1 3-ALKYNYL CARBOXAMIDES AS AEP MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2023-09-07 WO disclosed
EP-3683207-B1 N-ALKYLARYL-5-OXYARYL-OCTAHYDRO-CYCLOPENTA[C]PYRROLE NEGATIVE ALLOSTERIC MODULATORS OF NR2B CADENT THERAPEUTICS INC (US) 2021-12-29 EP disclosed