SCHEMBL2415544

SCHEMBL2415544

CN(Cc1cc(-c2cccnc2C#N)n(S(=O)(=O)c2ccc(F)cc2F)c1)C(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C2 P08235 2/20 0.36
HTR2C P28335 4/20 0.35
SLC6A4 P31645 4/20 0.35
HTR2A P28223 1/20 0.35
PPME1 Q9Y570 1/20 0.34
GRM4 Q14833 1/20 0.33
POLB P06746 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
PIK3C3 Q8NEB9 1/20 0.31
SQOR Q9Y6N5 1/20 0.31
ACLY P53396 1/20 0.31
LMNA P02545 1/20 0.30
IDH1 O75874 1/20 0.30
PLCG1 P19174 1/20 0.30
KDM2B Q8NHM5 1/20 0.30
KAT6A Q92794 1/20 0.30
KAT5 Q92993 1/20 0.30
AR P10275 1/20 0.30
PDE4A P27815 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2406675 0.93 HTR2C (0.34) NR3C2HTR2CSLC6A4HTR2APLCG1
SCHEMBL4410586 0.90 PPME1 (0.36) PPME1GRM4POLBCYP2C9CYP2C19
SCHEMBL2410588 0.89 HTR2C (0.32) NR3C2HTR2CSLC6A4HTR2APLCG1
SCHEMBL2414628 0.87 TACR1 (0.35) HTR2CSLC6A4PIK3C3SQORPLCG1
SCHEMBL2410003 0.87 HTR2C (0.34) HTR2CSLC6A4PLCG1KDM2B
SCHEMBL2412641 0.86 HTR2C (0.37) HTR2CSLC6A4LMNAPLCG1
SCHEMBL2409374 0.86 HTR2C (0.40) HTR2CSLC6A4HTR2APOLBKAT6A
SCHEMBL2409829 0.86 HTR2C (0.35) HTR2CSLC6A4PLCG1KAT6AKAT5
SCHEMBL2415547 0.84 PPME1 (0.35) NR3C2PPME1GRM4PIK3C3ACLY
SCHEMBL2416581 0.84 HTR2C (0.32) HTR2CSLC6A4PLCG1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed