SCHEMBL24174271

SCHEMBL24174271

Cc1cnc(OC(F)F)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.38
GRIN1 Q05586 6/20 0.36
GRIN2B Q13224 6/20 0.36
RXRA P19793 6/20 0.36
CYP3A4 P08684 2/20 0.34
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32
NOS2 P35228 1/20 0.32
SCN9A Q15858 2/20 0.31
LPAR1 Q92633 1/20 0.31
F2RL3 Q96RI0 3/20 0.31
PIK3CA P42336 1/20 0.31
ALDH1A1 P00352 1/20 0.30
TRPV4 Q9HBA0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24048533 0.85 ALOX5AP (0.36) CYP3A4CCR1CCR5CCR8NOS3
SCHEMBL17248014 0.82 NOS3 (0.42) GAAGRIN1GRIN2BRXRACCR1
SCHEMBL11918256 0.81 GAA (0.39) GAAGRIN1GRIN2BRXRACYP3A4
SCHEMBL16044313 0.79 GAA (0.35) GAAGRIN1GRIN2BRXRACCR1
SCHEMBL15599228 0.79 GAA (0.37) GAAGRIN1GRIN2BRXRASCN9A
SCHEMBL18371940 0.78 LPAR1 (0.37) GAAGRIN1GRIN2BRXRACYP3A4
SCHEMBL4150226 0.78 PIK3CA (0.45) CYP3A4CCR1CCR5CCR8NOS3
SCHEMBL22866537 0.77 RXRA (0.34) GAAGRIN1GRIN2BRXRATRPV4
SCHEMBL29560389 0.77 RXRA (0.34) GAAGRIN1GRIN2BRXRATRPV4
SCHEMBL25950819 0.77 ALDH1A1 (0.34) GAAGRIN1GRIN2BRXRAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022002097-A1 PYRAZOLO[1,5-A]PYRIDINE COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海艾力斯医药科技股份有限公司 2022-01-06 WO disclosed