SCHEMBL24176343

SCHEMBL24176343

Nc1c2c(nn1-c1ccncc1)CSC2

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 3/20 0.46
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
TSHR P16473 2/20 0.37
ALDH1A1 P00352 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HSD17B10 Q99714 1/20 0.37
MAPT P10636 1/20 0.36
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
SRC P12931 2/20 0.34
BRAF P15056 2/20 0.34
KDR P35968 2/20 0.34
LMNA P02545 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4882490 0.83 TSHR (0.49) KMT2AMEN1TSHRALDH1A1CYP1A2
SCHEMBL4881920 0.83 TP53 (0.47) ENPP2KMT2AMEN1TSHRMAPT
SCHEMBL24176322 0.83 ENPP2 (0.49) ENPP2KMT2AMEN1TSHRALDH1A1
SCHEMBL13858451 0.75 ALDH1A1 (0.42) KMT2AMEN1ALDH1A1HSD17B10SRC
SCHEMBL24176474 0.74 PDE2A (0.47) ENPP2LMNA
SCHEMBL12335147 0.63 SMN1; SMN2 (0.46) KMT2AMEN1ALDH1A1CYP1A2CYP2C19
SCHEMBL1073710 0.60 BRAF (0.43) ALDH1A1MAPTPOLBSRCBRAF
SCHEMBL1094177 0.60 PTGS2 (0.47) TSHRALDH1A1CYP1A2CYP3A4CYP2C19
SCHEMBL6086540 0.59 NPC1 (0.43) KMT2AMEN1TSHRALDH1A1CYP1A2
SCHEMBL13860846 0.58 NTRK1 (0.38) TSHRALDH1A1HSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022003377-A1 THIENO[3,4-C]PYRAZOL-3-YL ACETAMIDES AS AUTOTAXIN INHIBITORS UNI-PHARMA KLEON TSETIS PHARMACEUTICAL LABORATORIES S.A. (GR) 2022-01-06 WO disclosed