SCHEMBL24196864

SCHEMBL24196864

Cc1cccc(C#N)c1-c1ccc(S)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.48
HTR1A P08908 1/20 0.36
DRD2 P14416 1/20 0.36
HTR7 P34969 1/20 0.36
AR P10275 3/20 0.36
TRPV4 Q9HBA0 2/20 0.35
MAP4K1 Q92918 1/20 0.34
GRIA1 P42261 1/20 0.33
CACNG8 Q8WXS5 1/20 0.33
ALOX15 P16050 1/20 0.33
CASP1 P29466 1/20 0.33
CASP7 P55210 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
ESR2 Q92731 1/20 0.33
USP8 P40818 1/20 0.33
KLKB1 P03952 1/20 0.33
KDM4E B2RXH2 3/20 0.33
ALDH1A1 P00352 2/20 0.32
HPGD P15428 1/20 0.32
USP2 O75604 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4450143 0.83 TSHR (0.59) TSHRALOX15KDM4EALDH1A1HPGD
SCHEMBL21022697 0.80 TSHR (0.65) TSHRHTR1ADRD2HTR7AR
SCHEMBL26014276 0.80 GRIA1 (0.41) TSHRHTR7GRIA1CACNG8ALDH1A1
SCHEMBL21022696 0.78 TSHR (0.62) TSHRHTR1ADRD2HTR7AR
SCHEMBL24196851 0.78 TSHR (0.44) TSHRHTR1ADRD2HTR7AR
SCHEMBL30269804 0.77 CA2 (0.53) TSHR
SCHEMBL30270467 0.76 TSHR (0.42) TSHRGRIA1CACNG8USP8KDM4E
SCHEMBL942 0.75 TSHR (0.46) TSHRARESR2KDM4EALDH1A1
SCHEMBL24196740 0.75 AR (0.47) ARTRPV4EGLN2
SCHEMBL21189090 0.74 TSHR (0.47) TSHRAR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022008475-A1 INDOLE DERIVATIVES AND USES THEREOF FOR TREATING A CANCER UNIVERSITE CLAUDE BERNARD LYON 1 (FR) 2022-01-13 WO disclosed