SCHEMBL24202118

SCHEMBL24202118

C/C(=N\c1c(C)ncnc1N1CCc2cc(C)ccc21)NCCN(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 7/20 0.42
MKNK2 Q9HBH9 7/20 0.42
EIF4E P06730 4/20 0.42
SRD5A1 P18405 2/20 0.34
NOTUM Q6P988 1/20 0.34
PIK3CA P42336 1/20 0.34
MTOR P42345 1/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
CSF1R P07333 2/20 0.33
AURKA O14965 1/20 0.33
DAPK3 O43293 1/20 0.33
JAK2 O60674 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
ABL1 P00519 1/20 0.33
NTRK1 P04629 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23761571 0.95 MKNK1 (0.48) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL23761440 0.91 MKNK1 (0.53) MKNK1MKNK2EIF4ENOTUMPIK3CA
SCHEMBL24201711 0.89 MKNK1 (0.44) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL23761361 0.83 MKNK1 (0.39) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL24202017 0.80 NOTUM (0.41) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL23761552 0.79 MKNK1 (0.33) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL23761540 0.78 MKNK1 (0.36) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL24201720 0.77 KMT2A (0.40) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL24201658 0.74 SRD5A1 (0.41) MKNK1MKNK2EIF4ESRD5A1NOTUM
SCHEMBL23761414 0.72 SRD5A1 (0.45) MKNK1MKNK2EIF4ESRD5A1NOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3939981-A1 FUSED THIAZOLOPYRIMIDINE DERIVATIVES AS MNKS INHIBITORS LifeArc (GB) 2022-01-19 EP disclosed