SCHEMBL2420847

SCHEMBL2420847

NS(=O)(=O)c1cccc(C(F)(F)F)c1C1CC1

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.43
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
CA2 P00918 4/20 0.40
CA1 P00915 3/20 0.40
CA9 Q16790 3/20 0.40
CA5A P35218 2/20 0.40
PTGES2 Q9H7Z7 2/20 0.40
CA12 O43570 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA7 P43166 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
SCN9A Q15858 1/20 0.40
CHRNB2 P17787 1/20 0.40
CHRNA4 P43681 1/20 0.40
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4862690 0.84 PNMT (0.37) PNMTMEN1KMT2ACA2CA1
SCHEMBL30911354 0.82 PTGES2 (0.38) PNMTMEN1KMT2ACA2CA1
SCHEMBL29418255 0.75 MEN1 (0.56) MEN1KMT2ACA2CA1CA9
SCHEMBL302570 0.75 MEN1 (0.56) MEN1KMT2ACA2CA1CA9
SCHEMBL1336440 0.75 HTR2A (0.48) PNMTMEN1KMT2ASCN9ACHRNB2
SCHEMBL2777793 0.74 CA2 (0.47) MEN1KMT2ACA2CA1CA9
SCHEMBL2512044 0.74 CA2 (0.46) MEN1KMT2ACA2CA1CA9
SCHEMBL1659154 0.74 CHRNB2 (0.45) PNMTCHRNB2CHRNA4
SCHEMBL11685314 0.74 CA2 (0.50) MEN1KMT2ACA2CA1CA9
SCHEMBL2776294 0.74 CNR2 (0.41) MEN1KMT2ACA2CA1CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367790-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS Abbott Laboratories (US) 2011-09-28 EP claimed
WO-2010062927-A2 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2010-06-03 WO claimed
EP-2367790-A2 SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS Abbott Laboratories (US) 2011-09-28 EP disclosed
WO-2010062927-A2 NOVEL SUBSTITUTED OCTAHYDROCYCLOPENTA(C)PYRROL-4-AMINES AS CALCIUM CHANNEL BLOCKERS ABBOTT LABORATORIES (US) 2010-06-03 WO disclosed