SCHEMBL24247786

SCHEMBL24247786

CCC(=O)c1cnn2cc(OCCO)ccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.39
ROCK2 O75116 1/20 0.37
PDE2A O00408 4/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
GAA P10253 1/20 0.35
ROCK1 Q13464 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
ABL1 P00519 1/20 0.34
DRD2 P14416 1/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34
HTR2A P28223 1/20 0.34
DRD3 P35462 1/20 0.34
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21947201 0.86 HPGD (0.41) NR1I2SMN1; SMN2MEN1KMT2ANPC1
SCHEMBL20654123 0.85 ROCK2 (0.49) ROCK2PDE2ARAB9A
SCHEMBL20646745 0.85 ROCK2 (0.40) ROCK2PDE2ASMN1; SMN2MEN1KMT2A
SCHEMBL20646858 0.85 PDE2A (0.37) ROCK2PDE2ADRD2DRD1DRD4
SCHEMBL17437904 0.85 PRKAB2 (0.40) ROCK2SMN1; SMN2GAAROCK1NPC1
SCHEMBL20646991 0.84 ROCK2 (0.45) ROCK2PDE2A
SCHEMBL20647024 0.84 ROCK2 (0.40) ROCK2PDE2ASMN1; SMN2NPC1MAPT
SCHEMBL19997307 0.84 MEN1 (0.43) ROCK2PDE2ASMN1; SMN2MEN1KMT2A
SCHEMBL23889125 0.84 ROCK2 (0.36) ROCK2PDE2AJAK2JAK1TYK2
SCHEMBL21947322 0.83 KDM4E (0.49) SMN1; SMN2GAAMAPTDRD4HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3954681-A1 SPIROHEPTANE SALICYLAMIDES AND RELATED COMPOUNDS AS INHIBITORS OF ROCK Bristol-Myers Squibb Company (US) 2022-02-16 EP disclosed