SCHEMBL24253563

SCHEMBL24253563

CC(C)Cc1cc(F)c2c(c1)CCN(C)C2

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MAOA P21397 5/20 0.35
MAOB P27338 4/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
SLC6A4 P31645 1/20 0.34
HTR6 P50406 3/20 0.34
PTPN2 P17706 2/20 0.33
CHRNA7 P36544 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HRH1 P35367 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22993590 0.83 MAOA (0.38) MAOAMAOBCYP1A2CYP2D6SLC6A4
SCHEMBL22993218 0.75 MAOA (0.47) MAOAMAOBSLC6A4CHRNA7
SCHEMBL24253490 0.74 HRH3 (0.45) MAOAMAOBSLC6A4
SCHEMBL22993447 0.74 MAOA (0.41) MAOAMAOBCYP1A2CYP2D6SLC6A4
SCHEMBL25444508 0.74 MAOA (0.50) MAOAMAOBSLC6A4CHRNA7
SCHEMBL24253500 0.72 MAOA (0.45) MAOAMAOBCYP2D6SLC6A4CHRNA7
SCHEMBL22993619 0.71 MAOA (0.35) MAOAMAOBSLC6A4HTR6CHRNA7
SCHEMBL25121131 0.70 DRD2 (0.42) MAOAMAOBCYP1A2CYP2D6SLC6A4
SCHEMBL25091105 0.69 HTR2C (0.40) MAOAMAOBHTR6CHRNA7
SCHEMBL24253339 0.68 MAOA (0.37) MAOAMAOBSLC6A4HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230250080-A1 ENZYME INHIBITORS KALVISTA PHARMACEUTICALS LTD (GB) 2023-08-10 US disclosed
US-20230250080-A1 ENZYME INHIBITORS KALVISTA PHARMACEUTICALS LTD (GB) 2023-08-10 US disclosed
US-11613527-B2 Enzyme inhibitors KALVISTA PHARMACEUTICALS LIMITED (GB) 2023-03-28 US disclosed
US-20220048894-A1 ENZYME INHIBITORS KALVISTA PHARMACEUTICALS LIMITED (GB) 2022-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230250080-A1 ENZYME INHIBITORS SERPINB1, KLKB1, SERPINE1 MAOA 175/4885MAOB 71/4885CYP1A2 876/4885
US-11613527-B2 Enzyme inhibitors SERPINB1, KLKB1, SERPINE1 MAOA 175/4885MAOB 71/4885CYP1A2 876/4885
US-20220048894-A1 ENZYME INHIBITORS SERPINB1, KLKB1, SERPINE1 MAOA 175/4885MAOB 71/4885CYP1A2 876/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.