SCHEMBL24253949

SCHEMBL24253949

O=C1CCCC2(CCN(c3cc(OCC(F)(F)F)ncn3)CC2)N1c1ccc(Cl)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ELOVL1 Q9BW60 7/20 0.35
ACACB O00763 1/20 0.34
KCNH2 Q12809 2/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
LTC4S Q16873 1/20 0.33
PRKDC P78527 1/20 0.32
MGAT2 Q10469 1/20 0.32
AKT1 P31749 1/20 0.31
METTL3 Q86U44 1/20 0.31
PLA2G7 Q13093 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30494526 1.00 ELOVL1 (0.35) ELOVL1ACACBKCNH2HCRTR1HCRTR2
SCHEMBL24253624 0.92 ELOVL1 (0.37) ELOVL1ACACBKCNH2HCRTR1HCRTR2
SCHEMBL30423581 0.88 ELOVL1 (0.35) ELOVL1KCNH2HCRTR1HCRTR2LTC4S
SCHEMBL24253859 0.88 ELOVL1 (0.35) ELOVL1KCNH2HCRTR1HCRTR2LTC4S
SCHEMBL30494534 0.86 ABL1 (0.36) KCNH2HCRTR1HCRTR2LTC4SMGAT2
SCHEMBL24253872 0.86 ABL1 (0.36) KCNH2HCRTR1HCRTR2LTC4SMGAT2
SCHEMBL30494558 0.83 KCNH2 (0.34) KCNH2HCRTR1HCRTR2LTC4SPLA2G7
SCHEMBL24253842 0.83 KCNH2 (0.34) KCNH2HCRTR1HCRTR2LTC4SPLA2G7
SCHEMBL24253536 0.82 DPP4 (0.36) KCNH2HCRTR1HCRTR2LTC4SAKT1
SCHEMBL30494533 0.82 DPP4 (0.36) KCNH2HCRTR1HCRTR2LTC4SAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof NOVARTIS AG (CH) 2023-07-25 US disclosed
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof NOVARTIS AG (CH) 2023-07-25 US disclosed
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2022-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof REN, NR3C2, PKD1 ELOVL1 4619/4885ACACB 4122/4885KCNH2 282/4885
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF REN, NR3C2, PKD1 ELOVL1 4619/4885ACACB 4122/4885KCNH2 282/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.