SCHEMBL24253859

SCHEMBL24253859

O=C1CCCC2(CCN(c3cc(OCC(F)F)ncn3)CC2)N1c1ccc(Cl)c(F)c1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ELOVL1 Q9BW60 7/20 0.35
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
KCNH2 Q12809 1/20 0.33
LTC4S Q16873 1/20 0.33
AKT1 P31749 1/20 0.31
METTL3 Q86U44 1/20 0.31
CHRM4 P08173 1/20 0.31
MMP2 P08253 1/20 0.30
ADAMTS5 Q9UNA0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30423581 1.00 ELOVL1 (0.35) ELOVL1HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL24253949 0.88 ELOVL1 (0.35) ELOVL1HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL30494526 0.88 ELOVL1 (0.35) ELOVL1HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL30494533 0.82 DPP4 (0.36) HCRTR1HCRTR2KCNH2LTC4SAKT1
SCHEMBL24253536 0.82 DPP4 (0.36) HCRTR1HCRTR2KCNH2LTC4SAKT1
SCHEMBL24253624 0.80 ELOVL1 (0.37) ELOVL1HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL29048010 0.80 ELOVL1 (0.33) ELOVL1HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL30423985 0.78 HCRTR1 (0.35) HCRTR1HCRTR2KCNH2LTC4SMETTL3
SCHEMBL24253866 0.78 HCRTR1 (0.35) HCRTR1HCRTR2KCNH2LTC4SMETTL3
SCHEMBL24253726 0.77 DPP4 (0.36) HCRTR1HCRTR2KCNH2LTC4SMMP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof NOVARTIS AG (CH) 2023-07-25 US disclosed
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof NOVARTIS AG (CH) 2023-07-25 US disclosed
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF NOVARTIS INSTITUTES FOR BIOMEDICAL RESEARCH, INC. 2022-02-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11708366-B2 Heteroaryl substituted spiropiperidinyl derivatives and pharmaceutical uses thereof REN, NR3C2, PKD1 ELOVL1 4619/4885HCRTR1 2245/4885HCRTR2 3027/4885
US-20220048909-A1 HETEROARYL SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF REN, NR3C2, PKD1 ELOVL1 4619/4885HCRTR1 2245/4885HCRTR2 3027/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.