SCHEMBL24256963

SCHEMBL24256963

COc1ccc(CCNCc2sc3nc4c(c(C)c3c2N)CCC4)cc1OC

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.50
LMNA P02545 1/20 0.50
HPGD P15428 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
CYP1A2 P05177 2/20 0.43
BCHE P06276 2/20 0.43
ACHE P22303 2/20 0.43
ALDH1A1 P00352 2/20 0.43
KDM4E B2RXH2 1/20 0.43
GLA P06280 1/20 0.43
EEF2K O00418 1/20 0.42
MAPT P10636 1/20 0.41
ALOX15 P16050 1/20 0.40
CYP3A4 P08684 1/20 0.40
SMPD1 P17405 1/20 0.40
MTOR P42345 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24256678 0.82 LMNA (0.67) SMN1; SMN2LMNAHPGDKMT2AALDH1A1
SCHEMBL24256858 0.69 MTOR (0.63) SMN1; SMN2LMNAHPGDKMT2AALDH1A1
SCHEMBL24256612 0.66 MTOR (0.60) SMN1; SMN2LMNAHPGDKMT2AALDH1A1
SCHEMBL24256709 0.64 MTOR (0.61) SMN1; SMN2LMNAHPGDKMT2AALDH1A1
SCHEMBL30647980 0.64 DHFR (0.48) SMN1; SMN2LMNAHPGDCYP1A2BCHE
SCHEMBL7435099 0.64 ATM (0.76) SMN1; SMN2MEN1KMT2AALDH1A1KDM4E
SCHEMBL24256707 0.64 MTOR (0.58) SMN1; SMN2LMNAHPGDKMT2AALDH1A1
SCHEMBL9668420 0.64 ALDH1A1 (0.74) SMN1; SMN2LMNAMEN1KMT2AALDH1A1
Hydrochloric Acid SCHEMBL11808765 0.63 ATM (0.73) SMN1; SMN2MEN1KMT2AALDH1A1KDM4E
SCHEMBL11484160 0.63 ALDH1A1 (0.54) SMN1; SMN2LMNAMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022035806-A1 FUSED TRICYCLIC PYRIMIDINE-THIENO-PYRIDINE SMALL MOLECULE INHIBITORS OF UBIQUITIN-SPECIFIC PROTEASE 28 DANA-FARBER CANCER INSTITUTE, INC. (US) 2022-02-17 WO disclosed