SCHEMBL24258225

SCHEMBL24258225

Nc1cccc2c1CCCC21CCC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.35
CD44 P16070 2/20 0.34
SIGMAR1 Q99720 10/20 0.34
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
TP53 P04637 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
DRD2 P14416 1/20 0.33
TSHR P16473 1/20 0.33
NFKB1 P19838 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
MAPK1 P28482 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTR2B P41595 1/20 0.33
MTOR P42345 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24258173 0.96 KDM1A (0.35) KDM1ACD44SIGMAR1MEN1KMT2A
SCHEMBL21936668 0.92 CD44 (0.34) KDM1ACD44SIGMAR1MEN1KMT2A
SCHEMBL24258213 0.84 CD44 (0.36) KDM1ACD44SIGMAR1MEN1KMT2A
SCHEMBL15822259 0.79 KDM1A (0.41) KDM1ACD44MEN1KMT2ATP53
Hydrochloric Acid SCHEMBL15532871 0.78 KDM1A (0.40) KDM1ACD44MEN1KMT2ATP53
SCHEMBL21937081 0.77 SIGMAR1 (0.33) SIGMAR1MEN1KMT2ATP53CYP1A2
SCHEMBL24258207 0.74 CES2 (0.38) KDM1ACD44MEN1KMT2ATP53
SCHEMBL21937752 0.73 SIGMAR1 (0.35) KDM1ASIGMAR1MEN1KMT2ATP53
SCHEMBL21936942 0.73 PDE7A (0.36) SIGMAR1MEN1KMT2ATP53CYP1A2
SCHEMBL21937753 0.73 SIGMAR1 (0.33) SIGMAR1MEN1KMT2ATP53CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022036297-A1 NON-HYDRATED KETONE INHIBITORS OF NAV1.7 FOR THE TREATMENT OF PAIN SITEONE THERAPEUTICS, INC. (US) 2022-02-17 WO disclosed