SCHEMBL24259952

SCHEMBL24259952

CCCc1ccc(Sc2ccc3c(c2)C(C)(C)CCC3(C)C)cc1

nearest known ligand 0.64

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP26A1 O43174 6/20 0.64
RXRA P19793 8/20 0.57
RXRB P28702 6/20 0.57
RXRG P48443 6/20 0.57
RARB P10826 3/20 0.57
RARG P13631 3/20 0.57
CYP26B1 Q9NR63 7/20 0.45
CYP3A4 P08684 1/20 0.40
PPARG P37231 1/20 0.36
RARA P10276 1/20 0.35
LPL P06858 1/20 0.34
LIPG Q9Y5X9 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2897524 0.82 CYP26B1 (0.53) CYP26A1RXRARXRBRXRGRARB
SCHEMBL24259972 0.82 CYP26A1 (0.76) CYP26A1RXRARXRBRXRGRARB
SCHEMBL17911561 0.80 CYP26A1 (0.61) CYP26A1RXRARXRBRXRGRARB
SCHEMBL24259977 0.80 CYP26B1 (0.67) CYP26A1RXRARXRBRXRGRARB
SCHEMBL7759680 0.79 RXRA (0.69) CYP26A1RXRARXRBRXRGRARB
SCHEMBL24259981 0.79 CYP26A1 (0.57) CYP26A1RXRARXRBRXRGRARB
SCHEMBL17911573 0.78 CYP26A1 (1.00) CYP26A1RXRARXRBRXRGRARB
SCHEMBL17911584 0.76 CYP26A1 (0.67) CYP26A1RXRARXRBRXRGRARB
SCHEMBL29567511 0.76 CYP26A1 (0.67) CYP26A1RXRARXRBRXRGRARB
SCHEMBL577213 0.76 LPL (0.48) CYP3A4LPLLIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3044216-B1 NOVEL AND SPECIFIC INHIBITORS OF CYTOCHROME P450 26 RETINOIC ACID HYDROXYLASE UNIV WASHINGTON THROUGH ITS CENTER FOR COMMERCIALIZATION (US) 2022-02-23 EP disclosed