SCHEMBL24263131

SCHEMBL24263131

O=C(NC1CCc2n[nH]c(=O)cc2C1)c1ccc(Br)cc1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HDAC8 Q9BY41 3/20 0.45
CCNA2 P20248 5/20 0.42
CDK2 P24941 5/20 0.42
CCNA1 P78396 5/20 0.42
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
PAK1 Q13153 1/20 0.39
SMYD3 Q9H7B4 2/20 0.39
GAA P10253 1/20 0.38
SCN5A Q14524 1/20 0.38
SCN9A Q15858 1/20 0.38
SCN3A Q9NY46 1/20 0.38
NAMPT P43490 1/20 0.37
MMP2 P08253 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24263128 0.89 RAB9A (0.47) LMNAPAK1SMYD3GAANAMPT
SCHEMBL24263134 0.89 SMYD3 (0.39) HDAC8KMT2ASMYD3GAANAMPT
SCHEMBL24263090 0.89 NPC1 (0.47) HDAC8KMT2APAK1SMYD3GAA
SCHEMBL24263129 0.89 HDAC8 (0.48) HDAC8CCNA2CDK2CCNA1KMT2A
SCHEMBL24263127 0.88 MTNR1A (0.46) HDAC8CCNA2CDK2CCNA1KMT2A
SCHEMBL24263084 0.87 KMT2A (0.42) LMNAKMT2ASMYD3GAANAMPT
SCHEMBL24263197 0.86 TAOK1 (0.48) LMNAKMT2ASMYD3GAA
SCHEMBL24263089 0.86 KDM5A (0.40) HDAC8LMNAKMT2ASMYD3
SCHEMBL24263227 0.85 HDAC8 (0.42) HDAC8CCNA2CDK2CCNA1GAA
SCHEMBL24263079 0.84 TAOK1 (0.40) HDAC8SMYD3GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022040508-A1 COMPOUNDS AND METHODS FOR TREATING AUTOIMMUNE DISORDERS BY TARGETING HLA-DQ2 IMMUNOMOLECULAR THERAPEUTICS, INC. (US) 2022-02-24 WO disclosed