SCHEMBL24263271

SCHEMBL24263271

CNc1cc(Nc2cccc(C)n2)nn2c(C)cnc12

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TYK2 P29597 15/20 0.43
PDE4D Q08499 8/20 0.43
JAK2 O60674 2/20 0.41
JAK1 P23458 2/20 0.41
JAK3 P52333 2/20 0.41
MAP4K4 O95819 1/20 0.41
GSK3B P49841 1/20 0.41
GRM5 P41594 4/20 0.39
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24263473 0.84 TYK2 (0.53) TYK2PDE4DJAK2JAK1JAK3
SCHEMBL469978 0.75 TYK2 (0.39) TYK2PDE4D
SCHEMBL24263269 0.73 TYK2 (0.55) TYK2PDE4D
SCHEMBL24263303 0.72 TYK2 (0.55) TYK2PDE4D
SCHEMBL24263488 0.72 TYK2 (0.50) TYK2PDE4D
SCHEMBL24263537 0.69 TYK2 (0.70) TYK2
SCHEMBL24263560 0.69 TYK2 (0.38) TYK2PDE4D
SCHEMBL229747 0.69 RAB9A (0.59) GRM5KDR
SCHEMBL21571881 0.68 TYK2 (0.46) TYK2PDE4DJAK2JAK1JAK3
SCHEMBL20504498 0.67 TYK2 (0.58) TYK2PDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022037694-A1 A CLASS OF FIVE- AND SIX-MEMBERED HETEROCYCLIC COMPOUNDS AND USE THEREOF AS PROTEIN RECEPTOR KINASE INHIBITORS 轶诺(浙江)药业有限公司 2022-02-24 WO disclosed