SCHEMBL2426758

SCHEMBL2426758

C=CCCCCCN[C@H](C(=O)N1C[C@H](Oc2cc(-c3ccccc3)nc3cc(OC)c(C=C)cc23)C[C@H]1C(=O)OC)C1CCCCC1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DNMT1 P26358 2/20 0.34
EHMT2 Q96KQ7 2/20 0.34
CTSB P07858 2/20 0.33
PPP3CB P16298 1/20 0.33
ELANE P08246 1/20 0.31
KCNH2 Q12809 1/20 0.31
MAPT P10636 1/20 0.31
DHODH Q02127 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
EGFR P00533 1/20 0.30
HTR3E A5X5Y0 1/20 0.30
HTR3B O95264 1/20 0.30
HTR3A P46098 1/20 0.30
HTR3D Q70Z44 1/20 0.30
HTR3C Q8WXA8 1/20 0.30
HDAC1 Q13547 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4294855 0.96 DNMT1 (0.34) DNMT1EHMT2CTSBPPP3CBELANE
SCHEMBL2426760 0.86 DNMT1 (0.33) DNMT1EHMT2CTSBMAPTDHODH
SCHEMBL2429482 0.85 CYP3A4 (0.38) CTSBELANEKCNH2
SCHEMBL13026228 0.83 AAK1 (0.35) DNMT1EHMT2CTSBPPP3CBTDP1
SCHEMBL4298045 0.82 CYP3A4 (0.38) CTSBELANEKCNH2TDP1
SCHEMBL8221244 0.80 AAK1 (0.34) CTSBPPP3CB
SCHEMBL2894467 0.79 AAK1 (0.35) DNMT1EHMT2CTSBPPP3CB
SCHEMBL12963581 0.77 MEN1 (0.39) DHODHTDP1EGFRHTR3EHTR3B
SCHEMBL8213890 0.77 UCHL1 (0.43)
SCHEMBL13047543 0.77 CTSB (0.39) CTSBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041159-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2011-09-28 EP disclosed