SCHEMBL2429482

SCHEMBL2429482

C=CCCCCCN[C@H](C(=O)N1C[C@H](Oc2nccc3cc(OC)c(C=C)cc23)C[C@H]1C(=O)OC)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
ELANE P08246 1/20 0.35
KCNH2 Q12809 1/20 0.35
IRAK4 Q9NWZ3 5/20 0.32
CTSB P07858 1/20 0.31
MMP2 P08253 1/20 0.31
ANPEP P15144 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4298045 0.95 CYP3A4 (0.38) CYP3A4ELANEKCNH2IRAK4CTSB
SCHEMBL2426758 0.85 DNMT1 (0.34) ELANEKCNH2CTSB
SCHEMBL2429485 0.84 CYP3A4 (0.33) CYP3A4ELANEKCNH2IRAK4
SCHEMBL4294855 0.81 DNMT1 (0.34) ELANEKCNH2CTSB
SCHEMBL8195028 0.80 CYP3A4 (0.36) CYP3A4ELANEKCNH2IRAK4
SCHEMBL733229 0.80 CYP3A4 (0.39) CYP3A4ELANEKCNH2CTSB
SCHEMBL3624949 0.79 CYP3A4 (0.40) CYP3A4ELANEKCNH2IRAK4CTSB
SCHEMBL10081455 0.76 CYP3A4 (0.37) CYP3A4ELANEKCNH2IRAK4CTSB
SCHEMBL16318483 0.76 CYP3A4 (0.41) CYP3A4IRAK4CTSBMMP2ANPEP
SCHEMBL16318484 0.76 CYP3A4 (0.41) CYP3A4IRAK4CTSBMMP2ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041159-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2011-09-28 EP disclosed