SCHEMBL24282905

SCHEMBL24282905

CC#Cc1cccc(-n2ncc3cc(N4C(=O)CCC4c4ccccc4)ccc32)c1

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 9/20 0.39
HDAC1 Q13547 8/20 0.39
HDAC8 Q9BY41 7/20 0.39
HDAC5 Q9UQL6 5/20 0.39
TNKS O95271 2/20 0.37
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
NR3C1 P04150 3/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
HPGDS O60760 1/20 0.33
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32
MGLL Q99685 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21103720 0.89 IRAK4 (0.42) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL21103867 0.86 HDAC6 (0.46) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL21104025 0.82 PGR (0.47) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL24282907 0.82 PGR (0.47) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL24189829 0.81 NR3C1 (0.53) HDAC6HDAC1HDAC8HDAC5NR3C1
SCHEMBL25998434 0.79 NR3C1 (0.44) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL24282697 0.75 NR3C1 (0.47) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL24282864 0.75 NR3C1 (0.47) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL24283181 0.75 TNKS (0.47) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL24282791 0.75 TNKS (0.47) HDAC6HDAC1HDAC8HDAC5TNKS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728233-B1 SUBSTITUTED PYRROLIDINE AMIDES II GRUENENTHAL GMBH (DE) 2022-04-20 EP disclosed