SCHEMBL24282907

SCHEMBL24282907

N#Cc1ccc(-n2ncc3cc(N4C(=O)CCC4c4ccccc4)ccc32)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.47
HDAC6 Q9UBN7 6/20 0.42
HDAC1 Q13547 5/20 0.42
HDAC8 Q9BY41 5/20 0.42
HDAC5 Q9UQL6 3/20 0.42
TNKS O95271 4/20 0.40
NR3C1 P04150 4/20 0.39
CYP11B2 P19099 1/20 0.39
CYP19A1 P11511 2/20 0.35
CCNA2 P20248 1/20 0.35
CDK2 P24941 1/20 0.35
CCNA1 P78396 1/20 0.35
IDO1 P14902 1/20 0.34
TDO2 P48775 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21104025 1.00 PGR (0.47) PGRHDAC6HDAC1HDAC8HDAC5
SCHEMBL21103720 0.91 IRAK4 (0.42) PGRHDAC6HDAC1HDAC8HDAC5
SCHEMBL21103867 0.91 HDAC6 (0.46) PGRHDAC6HDAC1HDAC8HDAC5
SCHEMBL24189829 0.87 NR3C1 (0.53) PGRHDAC6HDAC1HDAC8HDAC5
SCHEMBL24282905 0.82 HDAC6 (0.39) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL22190386 0.81 HDAC6 (0.49) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL22201218 0.81 HDAC6 (0.49) HDAC6HDAC1HDAC8HDAC5TNKS
SCHEMBL25998434 0.81 NR3C1 (0.44) PGRHDAC6HDAC1HDAC8HDAC5
SCHEMBL24282697 0.81 NR3C1 (0.47) PGRHDAC6HDAC1HDAC8HDAC5
SCHEMBL24282864 0.81 NR3C1 (0.47) PGRHDAC6HDAC1HDAC8HDAC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3728233-B1 SUBSTITUTED PYRROLIDINE AMIDES II GRUENENTHAL GMBH (DE) 2022-04-20 EP disclosed