SCHEMBL2429485

SCHEMBL2429485

C=CCCCCCN[C@H](C(=O)N1C[C@H](Oc2nccc3cc(OC)c(C=C)cc23)C[C@@]1(C)C(=O)O)C1CCCCC1

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.33
IRAK4 Q9NWZ3 4/20 0.31
ELANE P08246 1/20 0.31
KCNH2 Q12809 1/20 0.31
GRM4 Q14833 1/20 0.30
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2426760 0.86 DNMT1 (0.33)
SCHEMBL4298045 0.85 CYP3A4 (0.38) CYP3A4IRAK4ELANEKCNH2KDM4E
SCHEMBL2429482 0.84 CYP3A4 (0.38) CYP3A4IRAK4ELANEKCNH2
SCHEMBL2427449 0.76 PIK3CD (0.38) CYP3A4IRAK4
SCHEMBL733230 0.76 CYP3A4 (0.33) CYP3A4ELANEKCNH2
SCHEMBL2427394 0.71 CYP3A4 (0.34) CYP3A4
SCHEMBL2426758 0.71 DNMT1 (0.34) ELANEKCNH2TDP1
SCHEMBL4294855 0.71 DNMT1 (0.34) ELANEKCNH2
SCHEMBL3624949 0.69 CYP3A4 (0.40) CYP3A4IRAK4ELANEKCNH2
SCHEMBL731548 0.69 CYP3A4 (0.33) CYP3A4ELANEKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041159-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2011-09-28 EP disclosed