SCHEMBL2427449

SCHEMBL2427449

C=Cc1cc2c(O[C@H]3CN(C(=O)OC(C)(C)C)[C@](C)(C(=O)O)C3)nccc2cc1OC

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.38
PIK3CA P42336 2/20 0.38
PIK3CB P42338 2/20 0.38
PIK3CG P48736 2/20 0.38
IRAK4 Q9NWZ3 12/20 0.34
CYP3A4 P08684 1/20 0.34
PDE4B Q07343 3/20 0.34
F13A1 P00488 1/20 0.33
TGM2 P21980 1/20 0.33
TGM1 P22735 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2430722 0.88 PIK3CD (0.38) PIK3CDPIK3CAPIK3CBPIK3CGIRAK4
SCHEMBL2428718 0.85 CYP3A4 (0.32) PIK3CDPIK3CAPIK3CBPIK3CGCYP3A4
SCHEMBL1072632 0.82 SMN1; SMN2 (0.36) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL3302407 0.81 GPR119 (0.36)
SCHEMBL2431240 0.81 RORC (0.35) PIK3CDPIK3CAPIK3CBPIK3CG
SCHEMBL1074490 0.81 CYP3A4 (0.40) PIK3CDPIK3CAPIK3CBPIK3CGIRAK4
SCHEMBL1074488 0.81 CYP3A4 (0.40) PIK3CDPIK3CAPIK3CBPIK3CGIRAK4
SCHEMBL1071024 0.80 PDE4B (0.33) PIK3CDPIK3CAPIK3CBPIK3CGPDE4B
SCHEMBL16318484 0.79 CYP3A4 (0.41) PIK3CDPIK3CAPIK3CBPIK3CGIRAK4
SCHEMBL16318483 0.79 CYP3A4 (0.41) PIK3CDPIK3CAPIK3CBPIK3CGIRAK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2041159-B1 MACROCYCLIC COMPOUNDS AS ANTIVIRAL AGENTS ANGELETTI P IST RICHERCHE BIO (IT) 2011-09-28 EP disclosed