SCHEMBL2430757

SCHEMBL2430757

O=C(CBr)OCCc1ccccc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.63
HCAR2 Q8TDS4 1/20 0.54
APP P05067 1/20 0.54
ESR1 P03372 1/20 0.53
ESR2 Q92731 1/20 0.53
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
AKR1B10 O60218 2/20 0.51
AKR1B1 P15121 2/20 0.51
TP53 P04637 1/20 0.51
GLA P06280 1/20 0.51
CYP3A4 P08684 1/20 0.51
HPGD P15428 1/20 0.51
TSHR P16473 1/20 0.51
MAPK1 P28482 1/20 0.51
HIF1A Q16665 1/20 0.51
HSD17B10 Q99714 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9361366 0.86 TDP1 (0.56) TDP1NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL451184 0.84 TDP1 (0.68) TDP1HCAR2APPESR1ESR2
SCHEMBL22832718 0.84 TDP1 (0.81) TDP1HCAR2APPESR1ESR2
SCHEMBL9367557 0.82 TDP1 (0.92) TDP1HCAR2APPESR1ESR2
SCHEMBL8890081 0.82 TDP1 (0.66) TDP1HCAR2APPESR1ESR2
SCHEMBL245747 0.82 ALDH1A1 (0.66) TDP1HCAR2APPESR1ESR2
SCHEMBL6025448 0.82 TDP1 (0.66) TDP1HCAR2APPESR1ESR2
SCHEMBL10731158 0.81 THRB (0.59) TDP1NPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL23760102 0.81 TDP1 (0.63) TDP1HCAR2APPESR1ESR2
SCHEMBL1960554 0.81 TDP1 (0.63) TDP1HCAR2APPESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105779130-A Method for preparing marigold volatile oil by fermentation and application of marigold volatile oil 湖北中烟工业有限责任公司 2016-07-20 CN disclosed
CN-102753542-B Substituted benzazepines as T0 LL-like receptor modulators VENTIRX PHARMACEUTICALS, INC. (US) 2016-01-20 CN disclosed
CN-104592016-A Efficient catalysis method for direct esterification and transesterification UNIV HUNAN 2015-05-06 CN disclosed
CN-101605775-B Substituted 3-phenyl-1-(phenylthienyl)propan-1-one and 3-phenyl-1-(phenylfuranyl)propan-1-one derivatives, and preparation and use of same GENFIT FR 2014-11-12 CN disclosed
US-20130046087-A1 Substituted Cyclodextrin Derivatives Useful As Intermediates For Producing Biologically Active Materials ARCARIOS BV (NL) 2013-02-21 US disclosed
EP-2550299-A2 Substituted cyclodextrin derivatives and process for their preparation Arcarios B.V. (NL) 2013-01-30 EP disclosed
CN-102834416-A Substituted cyclodextrin derivatives useful as intermediates for producing biologically active materials ARCARIOS BV 2012-12-19 CN disclosed
CN-102753542-A Substituted benzazepines as modulators of TOLL-like receptors VENTIRX PHARMACEUTICALS INC 2012-10-24 CN disclosed
WO-2011117317-A2 SUBSTITUTED CYCLODEXTRIN DERIVATIVES USEFUL AS INTERMEDIATES FOR PRODUCING BIOLOGICALLY ACTIVE MATERIALS ARCARIOS BV (NL) 2011-09-29 WO disclosed
CN-101605775-A 3-phenyl-1-(phenyl thienyl) third-1-ketone that replaces and derivative, preparation and the purposes of 3-phenyl-1-(benzofurane base) third-1-ketone GENFIT (FR) 2009-12-16 CN disclosed
WO-2008096128-A1 OXAZOLE AND THIAZOLE DERIVATIVES AND THEIR USES 2 ARGENTA DISCOVERY LTD (GB) 2008-08-14 WO disclosed
US-6562782-B1 Oligocycloalkanoids having a bacteriacidally effect; capable of binding lipids and/or endotoxins UNIVERSITY OF ROCHESTER 2003-05-13 US disclosed