SCHEMBL24315973

SCHEMBL24315973

CCc1ccccc1NC(C)CBr

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
POLB P06746 3/20 0.42
MAPT P10636 2/20 0.41
GAA P10253 2/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
GRIN2D O15399 1/20 0.38
GRIN3B O60391 1/20 0.38
GRIN1 Q05586 1/20 0.38
GRIN2A Q12879 1/20 0.38
GRIN2B Q13224 1/20 0.38
GRIN2C Q14957 1/20 0.38
GRIN3A Q8TCU5 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15325737 0.81 TAS1R3 (0.51) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL6023261 0.81 ALDH1A1 (0.47) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL8097565 0.80 ALDH1A1 (0.46) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL19038256 0.80 ALDH1A1 (0.46) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL30316736 0.80 ALDH1A1 (0.46) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL24635574 0.80 ALDH1A1 (0.41) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL17467884 0.79 POLB (0.46) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL12674140 0.79 KDM4E (0.46) ALDH1A1POLBMAPTGAATAS1R3
SCHEMBL9501212 0.78 ALDH1A1 (0.47) ALDH1A1POLBMAPTGAATAS1R3
Sulfuric Acid SCHEMBL9326018 0.75 ALDH1A1 (0.43) ALDH1A1POLBMAPTGAATAS1R3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3974423-A1 INDOLE DERIVATIVE-CONTAINING INHIBITOR, PREPARATION METHOD THEREFOR AND APPLICATION THEREOF Shanghai Hansoh Biomedical Co., Ltd. (CN) 2022-03-30 EP disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed