SCHEMBL24316016

SCHEMBL24316016

Sc1ccc(Cl)c(-c2cccc(Cl)c2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.41
ALOX5 P09917 1/20 0.40
DHFR P00374 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39
NUDT1 P36639 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
GAA P10253 1/20 0.37
RORB Q92753 1/20 0.37
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
ESR2 Q92731 1/20 0.37
NOTUM Q6P988 1/20 0.37
TP53 P04637 1/20 0.37
TSHR P16473 1/20 0.37
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3269842 0.84 TDO2 (0.46) TDO2ALOX5DHFRTAAR1NUDT1
SCHEMBL24315367 0.83 TDO2 (0.40) TDO2ALOX5DHFRTAAR1NUDT1
SCHEMBL10551642 0.82 CYP2A6 (0.54) ALOX5MEN1KMT2AESR2SMN1; SMN2
SCHEMBL21770705 0.77 ALDH1A1 (0.54) TDO2ALOX5DHFRTAAR1MEN1
SCHEMBL4450500 0.75 AHR (0.58) TDO2ALOX5DHFRTAAR1NUDT1
SCHEMBL29554995 0.75 AHR (0.58) TDO2ALOX5DHFRTAAR1NUDT1
SCHEMBL1520883 0.75 CYP2A6 (0.62) TDO2ALOX5DHFRTAAR1MEN1
SCHEMBL29464821 0.75 CYP2A6 (0.62) TDO2ALOX5DHFRTAAR1MEN1
SCHEMBL24315446 0.74 PRMT5 (0.44) ADORA2AADORA1
SCHEMBL16290690 0.73 CYP1A1 (0.50) KMT2ARORBNOTUMRELAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3619196-B1 2-{[2-(PHENYLOXYMETHYL)PYRIDIN-5-YL]OXY}-ETHANAMIN-DERIVATIVES AND RELATED COMPOUNDS AS PESTICIDES E.G. FOR CROP PROTECTION BAYER CROPSCIENCE AG (DE) 2022-03-30 EP disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed