SCHEMBL24316418

SCHEMBL24316418

COc1cc(O)cnc1OCc1ccc(C2CC2)cc1

nearest known ligand 0.41

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CSF1R P07333 17/20 0.41
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
NTRK1 P04629 1/20 0.38
TRPV6 Q9H1D0 1/20 0.38
QDPR P09417 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24316420 0.82 MAOB (0.45) CSF1R
SCHEMBL21327653 0.82 CSF1R (0.54) CSF1RNTRK1
SCHEMBL24316985 0.81 MRGPRX4 (0.49) CSF1R
SCHEMBL24316419 0.80 PDGFRB (0.49)
SCHEMBL29539254 0.78 EGFR (0.42) CSF1RKDM5AKDM4CKDM5BNTRK1
SCHEMBL24316790 0.78 EGFR (0.42) CSF1RKDM5AKDM4CKDM5BNTRK1
SCHEMBL24316988 0.77 CHRM4 (0.41) CSF1R
SCHEMBL27174564 0.74 ESR2 (0.42) KDM5AKDM4CKDM5B
SCHEMBL24316987 0.73 DHODH (0.38) CSF1R
SCHEMBL29859010 0.73 CSF1R (0.62) CSF1RNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022057895-A1 HETEROAROMATIC COMPOUNDS AND USES THEREOF HUTCHISON MEDIPHARMA LIMITED (CN) 2022-03-24 WO disclosed
US-9585884-B2 Pyrimidinone inhibitors of lipoprotein-associated phospholipase A2 AUSPEX PHARMACEUTICALS, INC. (US) 2017-03-07 US disclosed