SCHEMBL24316945

SCHEMBL24316945

Cc1cc(O)c(C)c(Cl)c1C

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.52
ALOX15 P16050 2/20 0.52
CHRM1 P11229 1/20 0.52
MAOA P21397 1/20 0.52
TBXA2R P21731 1/20 0.52
ADRA1A P35348 1/20 0.52
HTR2B P41595 1/20 0.52
ALDH1A1 P00352 4/20 0.50
MAPT P10636 3/20 0.50
GAA P10253 3/20 0.50
ACHE P22303 1/20 0.43
HPGD P15428 3/20 0.40
HSD17B10 Q99714 3/20 0.40
KDM4E B2RXH2 3/20 0.40
LMNA P02545 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
G6PD P11413 1/20 0.40
CYP2C9 P11712 1/20 0.40
PKM P14618 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2468038 0.84 CYP3A4 (0.52) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL7289170 0.84 ALDH1A1 (0.56) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL5589371 0.82 ALOX15 (0.50) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL14283744 0.82 MAPT (0.48) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL8724388 0.80 CYP3A4 (0.50) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL11055543 0.79 HSD17B10 (0.46) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL10820980 0.79 ALDH1A1 (0.50) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL8650668 0.79 ALDH1A1 (0.61) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL6722124 0.77 MAPT (0.54) CYP3A4ALOX15CHRM1MAOATBXA2R
SCHEMBL11038441 0.77 ALDH1A1 (0.48) CYP3A4ALOX15CHRM1MAOATBXA2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076285-A1 LACTAM COMPOUNDS AS Kv1.3 POTASSIUM SHAKER CHANNEL BLOCKERS D.E. SHAW RESEARCH, LLC (US) 2022-04-14 WO disclosed