SCHEMBL24320571

SCHEMBL24320571

CC(C)(C)OC(=O)N1CC=C(c2ccc(F)c(OCc3ccc(Cl)cc3F)c2)CC1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TLR7 Q9NYK1 1/20 0.47
NAMPT P43490 1/20 0.44
GPR119 Q8TDV5 2/20 0.44
KIT P10721 3/20 0.43
GRM5 P41594 6/20 0.43
GRM1 Q13255 6/20 0.43
CNR1 P21554 2/20 0.42
BRD4 O60885 1/20 0.42
ENPP2 Q13822 1/20 0.41
PDK4 Q16654 1/20 0.41
MKNK1 Q9BUB5 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30583903 0.92 TLR7 (0.47) TLR7NAMPTGPR119KITGRM5
SCHEMBL30453607 0.89 CNR1 (0.46) TLR7GPR119KITGRM5GRM1
SCHEMBL22391649 0.89 CNR1 (0.46) TLR7GPR119KITGRM5GRM1
SCHEMBL26914159 0.89 GPR119 (0.46) TLR7NAMPTGPR119KITGRM5
SCHEMBL24320715 0.88 KDM1A (0.45) TLR7NAMPTGPR119GRM5GRM1
SCHEMBL30284525 0.88 GRM5 (0.44) TLR7NAMPTGPR119KITGRM5
SCHEMBL22391814 0.88 GRM5 (0.44) TLR7NAMPTGPR119KITGRM5
SCHEMBL30583938 0.86 QDPR (0.45) TLR7NAMPTGPR119GRM5GRM1
SCHEMBL31306920 0.84 GRM1 (0.47) TLR7GPR119KITGRM5GRM1
SCHEMBL30583877 0.82 GRM5 (0.47) TLR7GPR119KITGRM5GRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230391760-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO, INC. 2023-12-07 US disclosed
WO-2022078407-A1 HETEROCYCLIC GLP-1 AGONISTS GASHERBRUM BIO, INC. (US) 2022-04-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230391760-A1 HETEROCYCLIC GLP-1 AGONISTS GLP1R, GIPR, GCGR TLR7 1125/4885NAMPT 2068/4885GPR119 11/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.