SCHEMBL24323797

SCHEMBL24323797

Cc1cccc(C)c1-c1cc(OC[C@H](N)CC2CC2)nc(NSc2cccc(C(=O)O)c2)n1

nearest known ligand 0.32

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LDHA P00338 2/20 0.32
LDHB P07195 2/20 0.32
NR1H4 Q96RI1 2/20 0.31
MEN1 O00255 1/20 0.31
NPC1 O15118 1/20 0.31
ALDH1A1 P00352 1/20 0.31
RAB9A P51151 1/20 0.31
KMT2A Q03164 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
SYK P43405 1/20 0.31
KDM4C Q9H3R0 1/20 0.30
VCP P55072 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24323721 0.97 LDHA (0.36) LDHALDHBKDM4C
SCHEMBL24298775 0.96 LDHA (0.35) LDHALDHBKDM4C
SCHEMBL24324172 0.96 LDHA (0.35) LDHALDHBKDM4C
SCHEMBL26569626 0.92
SCHEMBL24323694 0.92 LDHA (0.31) LDHALDHBNR1H4
SCHEMBL24298776 0.90
SCHEMBL24324641 0.89 CYP1A2 (0.31) LDHALDHBMEN1NPC1ALDH1A1
SCHEMBL26572133 0.89 GPR84 (0.37) MEN1ALDH1A1RAB9AKMT2ASMN1; SMN2
SCHEMBL24298810 0.87 AAK1 (0.34) LDHALDHBNR1H4MEN1NPC1
SCHEMBL22509294 0.87 AAK1 (0.34) LDHALDHBNR1H4MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed