SCHEMBL24324172

SCHEMBL24324172

Cc1cccc(C)c1-c1cc(OCC(N)CC2CCCCC2)nc(NSc2cccc(C(=O)O)c2)n1

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LDHA P00338 2/20 0.35
LDHB P07195 2/20 0.35
GUCY1B2 O75343 2/20 0.34
GUCY1A2 P33402 2/20 0.34
GUCY1A1 Q02108 2/20 0.34
GUCY1B1 Q02153 2/20 0.34
CDK1 P06493 1/20 0.32
CDK2 P24941 1/20 0.32
AKT1 P31749 2/20 0.32
EPHX1 P07099 1/20 0.32
KMO O15229 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
METAP2 P50579 2/20 0.31
PPM1D O15297 1/20 0.31
PTGER1 P34995 2/20 0.31
METAP1 P53582 1/20 0.31
GPR132 Q9UNW8 1/20 0.31
PRKCI P41743 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24298775 1.00 LDHA (0.35) LDHALDHBGUCY1B2GUCY1A2GUCY1A1
SCHEMBL24323721 0.99 LDHA (0.36) LDHALDHBGUCY1B2GUCY1A2GUCY1A1
SCHEMBL24323797 0.96 LDHA (0.32) LDHALDHBKDM4C
SCHEMBL26569626 0.90
SCHEMBL24298776 0.89
SCHEMBL26572133 0.89 GPR84 (0.37) KDM4CPTGER1
SCHEMBL24323694 0.88 LDHA (0.31) LDHALDHB
SCHEMBL24324641 0.87 CYP1A2 (0.31) LDHALDHB
SCHEMBL26576986 0.87 LDHA (0.35) LDHALDHBEPHX1
SCHEMBL24298880 0.86 MAPK8 (0.33) CDK1CDK2AKT1METAP2METAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076622-A2 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed