SCHEMBL24326511

SCHEMBL24326511

CC1=CC=C[C@H](C)[C@@H]1c1ccnc(N)n1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
CDK4 P11802 2/20 0.35
CDK2 P24941 2/20 0.35
CCNE1 P24864 1/20 0.35
HSP90AA1 P07900 3/20 0.33
AURKA O14965 1/20 0.33
PRKACA P17612 1/20 0.33
ADORA2A P29274 1/20 0.33
ROCK1 Q13464 3/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
MAP3K14 Q99558 1/20 0.31
HRH3 Q9Y5N1 1/20 0.30
CDK5 Q00535 1/20 0.30
CDK5R1 Q15078 1/20 0.30
NUDT1 P36639 1/20 0.30
HSP90AB1 P08238 1/20 0.30
PTK2 Q05397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24298898 0.77 HSP90AA1 (0.38) CDK2HSP90AA1NPC1RAB9AHRH3
SCHEMBL22783092 0.65 CYP3A4 (0.36)
SCHEMBL24786362 0.62 CASP1 (0.35) KDM4EALDH1A1MAPT
SCHEMBL1334584 0.62 ADORA2A (0.40) CDK4CDK2CCNE1HSP90AA1AURKA
SCHEMBL22919899 0.62 ALDH1A1 (0.35) ALDH1A1
SCHEMBL1334581 0.62 ADORA2A (0.40) CDK4CDK2CCNE1HSP90AA1AURKA
SCHEMBL2036795 0.62 ADORA2A (0.45) KDM4EALDH1A1CDK2HSP90AA1AURKA
Hydrochloric Acid SCHEMBL2018276 0.60 ADORA2A (0.44) KDM4EALDH1A1CDK2HSP90AA1AURKA
SCHEMBL29531700 0.60
SCHEMBL91470 0.60

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2022076625-A1 MODULATORS OF CYSTIC FIBROSIS TRANSMEMBRANE CONDUCTANCE REGULATOR VERTEX PHARMACEUTICALS INCORPORATED (US) 2022-04-14 WO disclosed